Standard InChI: InChI=1S/C19H32N8O5/c1-2-4-22-5-7-26(6-3-11(20)19(30)31)8-12-14(28)15(29)18(32-12)27-10-25-13-16(21)23-9-24-17(13)27/h9-12,14-15,18,22,28-29H,2-8,20H2,1H3,(H,30,31)(H2,21,23,24)/t11-,12+,14+,15+,18+/m0/s1
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2.Barsyte-Lovejoy, Dalia D and 32 more authors. 2014-09-02 (R)-PFI-2 is a potent and selective inhibitor of SETD7 methyltransferase activity in cells. [PMID:25136132]
3.Kaniskan, H Ümit; Konze, Kyle D and Jin, Jian. 2015-02-26 Selective inhibitors of protein methyltransferases. [PMID:25406853]
4.Takemoto, Yasushi Y and 16 more authors. 2016-04-28 Identification of Cyproheptadine as an Inhibitor of SET Domain Containing Lysine Methyltransferase 7/9 (Set7/9) That Regulates Estrogen-Dependent Transcription. [PMID:27088648]
5.Min, Wenjian and 10 more authors. 2020-04-01 Computational discovery and biological evaluation of novel inhibitors targeting histone-lysine N-methyltransferase SET7. [PMID:32088124]