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15. Gonzaga, Daniel Tadeu Gomes DTG and 16 more authors. 2017-10-20 1-Aryl-1H- and 2-aryl-2H-1,2,3-triazole derivatives blockade P2X7 receptor in vitro and inflammatory response in vivo. [PMID:28858765] |
16. Chrovian, Christa C CC and 17 more authors. 2018-01-11 A Dipolar Cycloaddition Reaction To Access 6-Methyl-4,5,6,7-tetrahydro-1H-[1,2,3]triazolo[4,5-c]pyridines Enables the Discovery Synthesis and Preclinical Profiling of a P2X7 Antagonist Clinical Candidate. [PMID:29211470] |
17. Homerin, Germain and 21 more authors. 2020-03-12 Pyroglutamide-Based P2X7 Receptor Antagonists Targeting Inflammatory Bowel Disease. [PMID:31525963] |
18. Bibic, Lucka; Herzig, Volker; King, Glenn F and Stokes, Leanne. 2019-09-27 Development of High-Throughput Fluorescent-Based Screens to Accelerate Discovery of P2X Inhibitors from Animal Venoms. [PMID:31532206] |
19. Calzaferri, Francesco and 7 more authors. 2021-02-25 Synthesis and Pharmacological Evaluation of Novel Non-nucleotide Purine Derivatives as P2X7 Antagonists for the Treatment of Neuroinflammation. [PMID:33560845] |