| 1. Wei J, Liu LL, Dong S, Li H, Tang D, Zhang Q, Xue QH, Gao JM.. (2016) Gabosines P and Q, new carbasugars from Streptomyces sp. and their α-glucosidase inhibitory activity., 26 (20): [PMID:27641469] [10.1016/j.bmcl.2016.09.021] |
| 2. Salar U, Taha M, Khan KM, Ismail NH, Imran S, Perveen S, Gul S, Wadood A.. (2016) Syntheses of new 3-thiazolyl coumarin derivatives, in vitro α-glucosidase inhibitory activity, and molecular modeling studies., 122 [PMID:27371923] [10.1016/j.ejmech.2016.06.037] |
| 3. Milella L, Milazzo S, De Leo M, Vera Saltos MB, Faraone I, Tuccinardi T, Lapillo M, De Tommasi N, Braca A.. (2016) α-Glucosidase and α-Amylase Inhibitors from Arcytophyllum thymifolium., 79 (8): [PMID:27509358] [10.1021/acs.jnatprod.6b00484] |
| 4. Wang G, Peng Z, Wang J, Li J, Li X.. (2016) Synthesis and biological evaluation of novel 2,4,5-triarylimidazole-1,2,3-triazole derivatives via click chemistry as α-glucosidase inhibitors., 26 (23): [PMID:27810241] [10.1016/j.bmcl.2016.10.057] |
| 5. Lee DY, Yang H, Kim HW, Sung SH.. (2017) New polyhydroxytriterpenoid derivatives from fruits of Terminalia chebula Retz. and their α-glucosidase and α-amylase inhibitory activity., 27 (1): [PMID:27890380] [10.1016/j.bmcl.2016.11.039] |
| 6. Sun H, Zhang Y, Ding W, Zhao X, Song X, Wang D, Li Y, Han K, Yang Y, Ma Y, Wang R, Wang D, Yu P.. (2016) Inhibitory activity evaluation and mechanistic studies of tetracyclic oxindole derivatives as α-glucosidase inhibitors., 123 [PMID:27487567] [10.1016/j.ejmech.2016.07.044] |
| 7. Wei M, Chai WM, Wang R, Yang Q, Deng Z, Peng Y.. (2017) Quinazolinone derivatives: Synthesis and comparison of inhibitory mechanisms on α-glucosidase., 25 (4): [PMID:28110817] [10.1016/j.bmc.2016.09.042] |
| 8. Wang K, Bao L, Ma K, Zhang J, Chen B, Han J, Ren J, Luo H, Liu H.. (2017) A novel class of α-glucosidase and HMG-CoA reductase inhibitors from Ganoderma leucocontextum and the anti-diabetic properties of ganomycin I in KK-Ay mice., 127 [PMID:27839787] [10.1016/j.ejmech.2016.11.015] |
| 9. Wang C, Guo L, Hao J, Wang L, Zhu W.. (2016) α-Glucosidase Inhibitors from the Marine-Derived Fungus Aspergillus flavipes HN4-13., 79 (11): [PMID:27933892] [10.1021/acs.jnatprod.6b00766] |
| 10. Verastegui-Omaña B, Rebollar-Ramos D, Pérez-Vásquez A, Martínez AL, Madariaga-Mazón A, Flores-Bocanegra L, Mata R.. (2017) α-Glucosidase Inhibitors from Malbranchea flavorosea., 80 (1): [PMID:28060505] [10.1021/acs.jnatprod.6b00977] |
| 11. Bisio A, De Mieri M, Milella L, Schito AM, Parricchi A, Russo D, Alfei S, Lapillo M, Tuccinardi T, Hamburger M, De Tommasi N.. (2017) Antibacterial and Hypoglycemic Diterpenoids from Salvia chamaedryoides., 80 (2): [PMID:28186413] [10.1021/acs.jnatprod.6b01053] |
| 12. Wang XL, Jiao FR, Yu M, Lin LB, Xiao J, Zhang Q, Wang L, Duan DZ, Xie G.. (2017) Constituents with potent α-glucosidase inhibitory activity from Pueraria lobata (Willd.) ohwi., 27 (9): [PMID:28343876] [10.1016/j.bmcl.2017.03.013] |
| 13. Kasturi S, Surarapu S, Uppalanchi S, Anireddy JS, Dwivedi S, Anantaraju HS, Perumal Y, Sigalapalli DK, Babu BN, Ethiraj KS.. (2017) Synthesis and α-glucosidase inhibition activity of dihydroxy pyrrolidines., 27 (12): [PMID:28495082] [10.1016/j.bmcl.2017.04.078] |
| 14. Morgan RE, van Staden CJ, Chen Y, Kalyanaraman N, Kalanzi J, Dunn RT, Afshari CA, Hamadeh HK.. (2013) A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development., 136 (1): [PMID:23956101] [10.1093/toxsci/kft176] |
| 15. Chen M, Suzuki A, Thakkar S, Yu K, Hu C, Tong W.. (2016) DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans., 21 (4): [PMID:26948801] [10.1016/j.drudis.2016.02.015] |
| 16. Jung HA, Paudel P, Seong SH, Min BS, Choi JS.. (2017) Structure-related protein tyrosine phosphatase 1B inhibition by naringenin derivatives., 27 (11): [PMID:28454670] [10.1016/j.bmcl.2017.04.054] |
| 17. Rangel-Grimaldo M, Rivero-Cruz I, Madariaga-Mazón A, Figueroa M, Mata R.. (2017) α-Glucosidase Inhibitors from Preussia minimoides ‡., 80 (3): [PMID:27673367] [10.1021/acs.jnatprod.6b00574] |
| 18. Wang G, Peng Z, Wang J, Li X, Li J.. (2017) Synthesis, in vitro evaluation and molecular docking studies of novel triazine-triazole derivatives as potential α-glucosidase inhibitors., 125 [PMID:27689725] [10.1016/j.ejmech.2016.09.067] |
| 19. Sun H, Ding W, Song X, Wang D, Chen M, Wang K, Zhang Y, Yuan P, Ma Y, Wang R, Dodd RH, Zhang Y, Lu K, Yu P.. (2017) Synthesis of 6-hydroxyaurone analogues and evaluation of their α-glucosidase inhibitory and glucose consumption-promoting activity: Development of highly active 5,6-disubstituted derivatives., 27 (15): [PMID:28651984] [10.1016/j.bmcl.2017.06.040] |
| 20. Zhang BW, Xing Y, Wen C, Yu XX, Sun WL, Xiu ZL, Dong YS.. (2017) Pentacyclic triterpenes as α-glucosidase and α-amylase inhibitors: Structure-activity relationships and the synergism with acarbose., 27 (22): [PMID:28964635] [10.1016/j.bmcl.2017.09.027] |
| 21. Nguyen CN, Trinh BTD, Tran TB, Nguyen LT, Jäger AK, Nguyen LD.. (2017) Anti-diabetic xanthones from the bark of Garcinia xanthochymus., 27 (15): [PMID:28624142] [10.1016/j.bmcl.2017.06.021] |
| 22. Xie Y, Yang Y, Li S, Xu Y, Lu W, Chen Z, Yang G, Li Y, Cao Y, Bian X.. (2017) Phenylsulfonylfuroxan NO-donor phenols: Synthesis and multifunctional activities evaluation., 25 (16): [PMID:28651914] [10.1016/j.bmc.2017.06.023] |
| 23. Flores-Bocanegra L, González-Andrade M, Bye R, Linares E, Mata R.. (2017) α-Glucosidase Inhibitors from Salvia circinata., 80 (5): [PMID:28422509] [10.1021/acs.jnatprod.7b00155] |
| 24. Pulvirenti L, Muccilli V, Cardullo N, Spatafora C, Tringali C.. (2017) Chemoenzymatic Synthesis and α-Glucosidase Inhibitory Activity of Dimeric Neolignans Inspired by Magnolol., 80 (5): [PMID:28497968] [10.1021/acs.jnatprod.7b00250] |
| 25. Prabha B, Neethu S, Krishnan SL, Sherin DR, Madhukrishnan M, Ananthakrishnan R, Rameshkumar KB, Manojkumar TK, Jayamurthy P, Radhakrishnan KV.. (2018) Antidiabetic potential of phytochemicals isolated from the stem bark of Myristica fatua Houtt. var. magnifica (Bedd.) Sinclair., 26 (12): [PMID:29789207] [10.1016/j.bmc.2018.05.020] |
| 26. Aydin G, Savran T, Baran Ş, Baran A.. (2018) Stereoselective synthesis of new rac-quercitols containing hydroxymethyl groups as glucosidase inhibitors., 28 (14): [PMID:29866516] [10.1016/j.bmcl.2018.05.034] |
| 27. Ibrar A, Shehzadi SA, Saeed F, Khan I.. (2018) Developing hybrid molecule therapeutics for diverse enzyme inhibitory action: Active role of coumarin-based structural leads in drug discovery., 26 (13): [PMID:30017112] [10.1016/j.bmc.2018.05.042] |
| 28. Gao E, Zhou ZQ, Zou J, Yu Y, Feng XL, Chen GD, He RR, Yao XS, Gao H.. (2017) Bioactive Asarone-Derived Phenylpropanoids from the Rhizome of Acorus tatarinowii Schott., 80 (11): [PMID:29116780] [10.1021/acs.jnatprod.7b00457] |
| 29. Wei Y, Wang C, Cheng Z, Tian X, Jia J, Cui Y, Feng L, Sun C, Zhang B, Ma X.. (2017) Heterodimeric Diterpenoids Isolated from Euphorbia ebracteolata Roots and Their Inhibitory Effects on α-Glucosidase., 80 (12): [PMID:29148766] [10.1021/acs.jnatprod.7b00595] |
| 30. Cai R, Wu Y, Chen S, Cui H, Liu Z, Li C, She Z.. (2018) Peniisocoumarins A-J: Isocoumarins from Penicillium commune QQF-3, an Endophytic Fungus of the Mangrove Plant Kandelia candel., 81 (6): [PMID:29792702] [10.1021/acs.jnatprod.7b01018] |
| 31. Adib M, Peytam F, Rahmanian-Jazi M, Mahernia S, Bijanzadeh HR, Jahani M, Mohammadi-Khanaposhtani M, Imanparast S, Faramarzi MA, Mahdavi M, Larijani B.. (2018) New 6-amino-pyrido[2,3-d]pyrimidine-2,4-diones as novel agents to treat type 2 diabetes: A simple and efficient synthesis, α-glucosidase inhibition, molecular modeling and kinetic study., 155 [PMID:29902721] [10.1016/j.ejmech.2018.05.046] |
| 32. Wang G, Chen M, Qiu J, Xie Z, Cao A.. (2018) Synthesis, in vitro α-glucosidase inhibitory activity and docking studies of novel chromone-isatin derivatives., 28 (2): [PMID:29208524] [10.1016/j.bmcl.2017.11.047] |
| 33. Wang K, Bao L, Zhou N, Zhang J, Liao M, Zheng Z, Wang Y, Liu C, Wang J, Wang L, Wang W, Liu S, Liu H.. (2018) Structural Modification of Natural Product Ganomycin I Leading to Discovery of a α-Glucosidase and HMG-CoA Reductase Dual Inhibitor Improving Obesity and Metabolic Dysfunction in Vivo., 61 (8): [PMID:29634260] [10.1021/acs.jmedchem.8b00107] |
| 34. Choi J, Yoon KD, Kim J.. (2018) Chemical constituents from Taraxacum officinale and their α-glucosidase inhibitory activities., 28 (3): [PMID:29254644] [10.1016/j.bmcl.2017.12.014] |
| 35. Sun Y, Liu J, Li L, Gong C, Wang S, Yang F, Hua H, Lin H.. (2018) New butenolide derivatives from the marine sponge-derived fungus Aspergillus terreus., 28 (3): [PMID:29295795] [10.1016/j.bmcl.2017.12.049] |
| 36. Dang PH, Nguyen HX, Duong TTT, Tran TKT, Nguyen PT, Vu TKT, Vuong HC, Phan NHT, Nguyen MTT, Nguyen NT, Awale S.. (2017) α-Glucosidase Inhibitory and Cytotoxic Taxane Diterpenoids from the Stem Bark of Taxus wallichiana., 80 (4): [PMID:28240909] [10.1021/acs.jnatprod.7b00006] |
| 37. Dang PH, Nguyen HX, Nguyen HHT, Vo TD, Le TH, Phan THN, Nguyen MTT, Nguyen NT.. (2017) Lignans from the Roots of Taxus wallichiana and Their α-Glucosidase Inhibitory Activities., 80 (6): [PMID:28581744] [10.1021/acs.jnatprod.7b00171] |
| 38. Ali F, Khan KM, Salar U, Taha M, Ismail NH, Wadood A, Riaz M, Perveen S.. (2017) Hydrazinyl arylthiazole based pyridine scaffolds: Synthesis, structural characterization, in vitro α-glucosidase inhibitory activity, and in silico studies., 138 [PMID:28672278] [10.1016/j.ejmech.2017.06.041] |
| 39. Ren J, Ding SS, Zhu A, Cao F, Zhu HJ.. (2017) Bioactive Azaphilone Derivatives from the Fungus Talaromyces aculeatus., 80 (8): [PMID:28749670] [10.1021/acs.jnatprod.7b00032] |
| 40. Zhang XQ, Mou XF, Mao N, Hao JJ, Liu M, Zheng JY, Wang CY, Gu YC, Shao CL.. (2018) Design, semisynthesis, α-glucosidase inhibitory, cytotoxic, and antibacterial activities of p-terphenyl derivatives., 146 [PMID:29407953] [10.1016/j.ejmech.2018.01.057] |
| 41. Kasturi SP, Surarapu S, Uppalanchi S, Dwivedi S, Yogeeswari P, Sigalapalli DK, Bathini NB, Ethiraj KS, Anireddy JS.. (2018) Synthesis, molecular modeling and evaluation of α-glucosidase inhibition activity of 3,4-dihydroxy piperidines., 150 [PMID:29518717] [10.1016/j.ejmech.2018.02.072] |
| 42. Adegboye AA, Khan KM, Salar U, Aboaba SA, Kanwal, Chigurupati S, Fatima I, Taha M, Wadood A, Mohammad JI, Khan H, Perveen S.. (2018) 2-Aryl benzimidazoles: Synthesis, In vitro α-amylase inhibitory activity, and molecular docking study., 150 [PMID:29533872] [10.1016/j.ejmech.2018.03.011] |
| 43. Karakılıç E, Durmuş S, Sevmezler S, Şahin O, Baran A.. (2018) Regio- and stereospecific synthesis of rac-carbasugar-based cyclohexane pentols; Investigations of their α- and β-glucosidase inhibitions., 26 (14): [PMID:30031655] [10.1016/j.bmc.2018.07.021] |
| 44. Luthra T, Naga Lalitha K, Agarwal R, Uma A, Sen S.. (2018) Design, synthesis and in vitro study of densely functionalized oxindoles as potent α-glucosidase inhibitors., 26 (18): [PMID:30153956] [10.1016/j.bmc.2018.08.022] |
| 45. Taha M, Irshad M, Imran S, Chigurupati S, Selvaraj M, Rahim F, Ismail NH, Nawaz F, Khan KM.. (2017) Synthesis of piperazine sulfonamide analogs as diabetic-II inhibitors and their molecular docking study., 141 [PMID:29102178] [10.1016/j.ejmech.2017.10.028] |
| 46. Kumar P, Duhan M, Kadyan K, Sindhu J, Kumar S, Sharma H.. (2017) Synthesis of novel inhibitors of α-amylase based on the thiazolidine-4-one skeleton containing a pyrazole moiety and their configurational studies., 8 (7): [PMID:30108858] [10.1039/C7MD00080D] |
| 47. Kasturi S, Surarapu S, Bathoju CC, Uppalanchi S, Dwivedi S, Perumal Y, Sigalapalli DK, Babu BN, Ethiraj KS, Anireddy JS.. (2017) Synthesis, molecular modeling and biological evaluation of aza-flavanones as α-glucosidase inhibitors., 8 (8): [PMID:30108873] [10.1039/C7MD00162B] |
| 48. Wang GC, Peng YP, Xie ZZ, Wang J, Chen M.. (2017) Synthesis, α-glucosidase inhibition and molecular docking studies of novel thiazolidine-2,4-dione or rhodanine derivatives., 8 (7): [PMID:30108859] [10.1039/C7MD00173H] |
| 49. Yousuf S, Khan KM, Salar U, Chigurupati S, Muhammad MT, Wadood A, Aldubayan M, Vijayan V, Riaz M, Perveen S.. (2018) 2'-Aryl and 4'-arylidene substituted pyrazolones: As potential α-amylase inhibitors., 159 [PMID:30268823] [10.1016/j.ejmech.2018.09.052] |
| 50. Dhameja M, Gupta P.. (2019) Synthetic heterocyclic candidates as promising α-glucosidase inhibitors: An overview., 176 [PMID:31112894] [10.1016/j.ejmech.2019.04.025] |
| 51. Spasov AA, Babkov DA, Osipov DV, Klochkov VG, Prilepskaya DR, Demidov MR, Osyanin VA, Klimochkin YN.. (2019) Synthesis, in vitro and in vivo evaluation of 2-aryl-4H-chromene and 3-aryl-1H-benzo[f]chromene derivatives as novel α-glucosidase inhibitors., 29 (1): [PMID:30340897] [10.1016/j.bmcl.2018.10.018] |
| 52. Li T, Kongstad KT, Staerk D.. (2019) Identification of α-Glucosidase Inhibitors in Machilus litseifolia by Combined Use of High-Resolution α-Glucosidase Inhibition Profiling and HPLC-PDA-HRMS-SPE-NMR., 82 (2): [PMID:30668111] [10.1021/acs.jnatprod.8b00609] |
| 53. Raksat A, Phukhatmuen P, Yang J, Maneerat W, Charoensup R, Andersen RJ, Wang YA, Pyne SG, Laphookhieo S.. (2020) Phloroglucinol Benzophenones and Xanthones from the Leaves of Garcinia cowa and Their Nitric Oxide Production and α-Glucosidase Inhibitory Activities., 83 (1): [PMID:31860303] [10.1021/acs.jnatprod.9b00849] |
| 54. Olanipekun BE, Ponnapalli MG, Shaik K, Nanubolu JB, Kommalapati VK, Tangutur AD.. (2020) α-Glucosidase Inhibitory Isomeric Corniculatolides from the Stems of the Indian Mangrove Plant, Xylocarpus granatum., 83 (1): [PMID:31895570] [10.1021/acs.jnatprod.9b00414] |
| 55. Saeedi M, Mohammadi-Khanaposhtani M, Asgari MS, Eghbalnejad N, Imanparast S, Faramarzi MA, Larijani B, Mahdavi M, Akbarzadeh T.. (2019) Design, synthesis, in vitro, and in silico studies of novel diarylimidazole-1,2,3-triazole hybrids as potent α-glucosidase inhibitors., 27 (23): [PMID:31679980] [10.1016/j.bmc.2019.115148] |
| 56. Chen M, Wang K, Zhang Y, Zhang M, Ma Y, Sun H, Jin Z, Zheng H, Jiang H, Yu P, Zhang Y, Sun H.. (2019) New insights into the biological activities of Chrysanthemum morifolium: Natural flavonoids alleviate diabetes by targeting α-glucosidase and the PTP-1B signaling pathway., 178 [PMID:31176093] [10.1016/j.ejmech.2019.05.083] |
| 57. Garg V, Maurya RK, Thanikachalam PV, Bansal G, Monga V.. (2019) An insight into the medicinal perspective of synthetic analogs of indole: A review., 180 [PMID:31344615] [10.1016/j.ejmech.2019.07.019] |
| 58. Santilli AD, Russell JT, Triplett EW, Whitehead KJ, Whitehead DC.. (2019) Non-lethal growth inhibition by arresting the starch utilization system of clinically relevant human isolates of Bacteroides dorei., 10 (11): [PMID:32280435] [10.1039/C9MD00301K] |
| 59. Liao HX, Zheng CJ, Huang GL, Mei RQ, Nong XH, Shao TM, Chen GY, Wang CY.. (2019) Bioactive Polyketide Derivatives from the Mangrove-Derived Fungus Daldinia eschscholtzii HJ004., 82 (8): [PMID:31373815] [10.1021/acs.jnatprod.9b00241] |
| 60. Meena SN, Kumar U, Naik MM, Ghadi SC, Tilve SG.. (2019) α-Glucosidase inhibition activity and in silico study of 2-(benzo[d][1,3]dioxol-5-yl)-4H-chromen-4-one, a synthetic derivative of flavone., 27 (12): [PMID:30594450] [10.1016/j.bmc.2018.12.021] |
| 61. Luo HY, Guo RX, Yu XK, Zhang X, Lu YQ, Wu HW, Tang LY, Wang ZJ.. (2019) Chemical constituents from the seeds of Cassia obtusefolia and their in vitro α-glucosidase inhibitory and antioxidant activities., 29 (13): [PMID:31078411] [10.1016/j.bmcl.2019.05.002] |
| 62. Taha M, Sultan S, Imran S, Rahim F, Zaman K, Wadood A, Ur Rehman A, Uddin N, Mohammed Khan K.. (2019) Synthesis of quinoline derivatives as diabetic II inhibitors and molecular docking studies., 27 (18): [PMID:31378594] [10.1016/j.bmc.2019.07.035] |
| 63. Shivanagoudra SR, Perera WH, Perez JL, Athrey G, Sun Y, Wu CS, Jayaprakasha GK, Patil BS.. (2019) In vitro and in silico elucidation of antidiabetic and anti-inflammatory activities of bioactive compounds from Momordica charantia L., 27 (14): [PMID:31196754] [10.1016/j.bmc.2019.05.035] |
| 64. Pathania S, Narang RK, Rawal RK.. (2019) Role of sulphur-heterocycles in medicinal chemistry: An update., 180 [PMID:31330449] [10.1016/j.ejmech.2019.07.043] |
| 65. Hameed S, Kanwal, Seraj F, Rafique R, Chigurupati S, Wadood A, Rehman AU, Venugopal V, Salar U, Taha M, Khan KM.. (2019) Synthesis of benzotriazoles derivatives and their dual potential as α-amylase and α-glucosidase inhibitors in vitro: Structure-activity relationship, molecular docking, and kinetic studies., 183 [PMID:31514061] [10.1016/j.ejmech.2019.111677] |
| 66. Suthiphasilp V, Maneerat W, Andersen RJ, Phukhatmuen P, Pyne SG, Laphookhieo S.. (2019) Dasymaschalolactams A-E, Aristolactams from a Twig Extract of Dasymaschalon dasymaschalum., 82 (11): [PMID:31661271] [10.1021/acs.jnatprod.9b00506] |
| 67. Adib M, Peytam F, Shourgeshty R, Mohammadi-Khanaposhtani M, Jahani M, Imanparast S, Faramarzi MA, Larijani B, Moghadamnia AA, Esfahani EN, Bandarian F, Mahdavi M.. (2019) Design and synthesis of new fused carbazole-imidazole derivatives as anti-diabetic agents: In vitro α-glucosidase inhibition, kinetic, and in silico studies., 29 (5): [PMID:30661823] [10.1016/j.bmcl.2019.01.012] |
| 68. Zhong YY, Chen HS, Wu PP, Zhang BJ, Yang Y, Zhu QY, Zhang CG, Zhao SQ.. (2019) Synthesis and biological evaluation of novel oleanolic acid analogues as potential α-glucosidase inhibitors., 164 [PMID:30677669] [10.1016/j.ejmech.2018.12.046] |
| 69. Cardullo N, Catinella G, Floresta G, Muccilli V, Rosselli S, Rescifina A, Bruno M, Tringali C.. (2019) Synthesis of Rosmarinic Acid Amides as Antioxidative and Hypoglycemic Agents., 82 (3): [PMID:30785286] [10.1021/acs.jnatprod.8b01002] |
| 70. Meesakul P, Richardson C, Pyne SG, Laphookhieo S.. (2019) α-Glucosidase Inhibitory Flavonoids and Oxepinones from the Leaf and Twig Extracts of Desmos cochinchinensis., 82 (4): [PMID:30835120] [10.1021/acs.jnatprod.8b00581] |
| 71. Thao NP, Luyen BT, Vinh le B, Lee JY, Kwon YI, Kim YH.. (2016) Rat intestinal sucrase inhibited by minor constituents from the leaves and twigs of Archidendron clypearia (Jack.) Nielsen., 26 (17): [PMID:27481560] [10.1016/j.bmcl.2016.07.044] |
| 72. Özil M, Emirik M, Beldüz A, Ülker S.. (2016) Molecular docking studies and synthesis of novel bisbenzimidazole derivatives as inhibitors of α-glucosidase., 24 (21): [PMID:27576293] [10.1016/j.bmc.2016.08.024] |
| 73. Maria Kuzikov, Elisa Costanzi, Jeanette Reinshagen, Francesca Esposito, Laura Vangeel, Markus Wolf, Bernhard Ellinger, Carsten Claussen, Gerd Geisslinger, Angela Corona, Daniela Iaconis, Carmine Talarico, Candida Manelfi, Rolando Cannalire, Giulia Rossetti, Jonas Gossen, Simone Albani, Francesco Musiani, Katja Herzog, Yang Ye, Barbara Giabbai, Nicola Demitri, Dirk Jochmans, Steven De Jonghe, Jasper Rymenants, Vincenzo Summa, Enzo Tramontano, Andrea R. Beccari, Pieter Leyssen, Paola Storici, Johan Neyts, Philip Gribbon, and Andrea Zaliani. (2020) Identification of inhibitors of SARS-Cov2 M-Pro enzymatic activity using a small molecule repurposing screen, [10.6019/CHEMBL4495564] |
| 74. Andrea Zaliani, Laura Vangeel, Jeanette Reinshagen, Daniela Iaconis, Maria Kuzikov, Oliver Keminer, Markus Wolf, Bernhard Ellinger, Francesca Esposito, Angela Corona, Enzo Tramontano, Candida Manelfi, Katja Herzog, Dirk Jochmans, Steven De Jonghe, Winston Chiu, Thibault Francken, Joost Schepers, Caroline Collard, Kayvan Abbasi, Carsten Claussen , Vincenzo Summa, Andrea R. Beccari, Johan Neyts, Philip Gribbon and Pieter Leyssen. (2020) Cytopathic SARS-Cov2 screening on VERO-E6 cells in a large repurposing effort, [10.6019/CHEMBL4495565] |
| 75. Johannes Zuegg, Alysha Elliott, Maite Amado, Emma Cowie, Ali Hinton, Geraldine Kaeslin, Angela Kavanagh, Anne Kunert, Gabriell Lowe, Soumya Ramu, Janet Reid, Robin Trauer, Mathilde Desselle, Ruth Neale, Karl Hansford, Mark Blascovich, Matthew Cooper. CO-ADD screening of NIH (USA) - Clinical Collection, [10.6019/CHEMBL4513141] |
| 76. Yang F, Zhu W, Sun S, Ai Q, Edirisuriya P, Zhou K.. (2020) Isolation and Structural Characterization of Specific Bacterial β-Glucuronidase Inhibitors from Noni (Morinda citrifolia) Fruits., 83 (4): [PMID:32083868] [10.1021/acs.jnatprod.9b00279] |
| 77. Fan JR, Kuang Y, Dong ZY, Yi Y, Zhou YX, Li B, Qiao X, Ye M.. (2020) Prenylated Phenolic Compounds from the Aerial Parts of Glycyrrhiza uralensis as PTP1B and α-Glucosidase Inhibitors., 83 (4): [PMID:32196343] [10.1021/acs.jnatprod.9b00262] |
| 78. Rangel-Grimaldo M, Macías-Rubalcava ML, González-Andrade M, Raja H, Figueroa M, Mata R.. (2020) α-Glucosidase and Protein Tyrosine Phosphatase 1B Inhibitors from Malbranchea circinata., 83 (3): [PMID:31898904] [10.1021/acs.jnatprod.9b01108] |
| 79. Ahn JH, Park Y, Yeon SW, Jo YH, Han YK, Turk A, Ryu SH, Hwang BY, Lee KY, Lee MK.. (2020) Phenylpropanoid-Conjugated Triterpenoids from the Leaves of Actinidia arguta and Their Inhibitory Activity on α-Glucosidase., 83 (5): [PMID:32315181] [10.1021/acs.jnatprod.9b00643] |
| 80. Dowarah J, Singh VP.. (2020) Anti-diabetic drugs recent approaches and advancements., 28 (5): [PMID:32008883] [10.1016/j.bmc.2019.115263] |
| 81. Yeye EO, Kanwal, Mohammed Khan K, Chigurupati S, Wadood A, Ur Rehman A, Perveen S, Kannan Maharajan M, Shamim S, Hameed S, Aboaba SA, Taha M.. (2020) Syntheses, in vitro α-amylase and α-glucosidase dual inhibitory activities of 4-amino-1,2,4-triazole derivatives their molecular docking and kinetic studies., 28 (11): [PMID:32327353] [10.1016/j.bmc.2020.115467] |
| 82. Xie YD, Liu JP, Wang W, Shi YH, Wang XP, Sun M, Xu XY, Li N.. (2020) 3,4-Dihydroxyphenethyl nitrate with nitric oxide releasing, antioxidant, hypoglycemic and hypolipidemic effects., 30 (15): [PMID:32527456] [10.1016/j.bmcl.2020.127277] |
| 83. Hao L, Ma Y, Zhao L, Zhang Y, Zhang X, Ma Y, Dodd RH, Sun H, Yu P.. (2020) Synthesis of tetracyclic oxindoles and evaluation of their α-glucosidase inhibitory and glucose consumption-promoting activity., 30 (14): [PMID:32527562] [10.1016/j.bmcl.2020.127264] |
| 84. Yang XT, Geng CA, Li TZ, Deng ZT, Chen JJ.. (2020) Synthesis and biological evaluation of chepraecoxin A derivatives as α-glucosidase inhibitors., 30 (8): [PMID:32067867] [10.1016/j.bmcl.2020.127020] |
| 85. Ha MT, Kim M, Kim CS, Park SE, Kim JA, Woo MH, Choi JS, Min BS.. (2020) Tetra-aryl cyclobutane and stilbenes from the rhizomes of Rheum undulatum and their α-glucosidase inhibitory activity: Biological evaluation, kinetic analysis, and molecular docking simulation., 30 (8): [PMID:32111435] [10.1016/j.bmcl.2020.127049] |
| 86. Suthiphasilp V, Maneerat W, Rujanapun N, Duangyod T, Charoensup R, Deachathai S, Andersen RJ, Patrick BO, Pyne SG, Laphookhieo S.. (2020) α-Glucosidase inhibitory and nitric oxide production inhibitory activities of alkaloids isolated from a twig extract of Polyalthia cinnamomea., 28 (10): [PMID:32247751] [10.1016/j.bmc.2020.115462] |
| 87. Solangi M,Kanwal null,Mohammed Khan K,Saleem F,Hameed S,Iqbal J,Shafique Z,Qureshi U,Ul-Haq Z,Taha M,Perveen S. (2020) Indole acrylonitriles as potential anti-hyperglycemic agents: Synthesis, α-glucosidase inhibitory activity and molecular docking studies., 28 (21.0): [PMID:33065441] [10.1016/j.bmc.2020.115605] |
| 88. Takashima K,Sakano M,Kinouchi E,Nakamura S,Marumoto S,Ishikawa F,Ninomiya K,Nakanishi I,Morikawa T,Tanabe G. (2021) Elongation of the side chain by linear alkyl groups increases the potency of salacinol, a potent α-glucosidase inhibitor from the Ayurvedic traditional medicine "Salacia," against human intestinal maltase., 33 [PMID:33347966] [10.1016/j.bmcl.2020.127751] |
| 89. Madasu C,Karri S,Sangaraju R,Sistla R,Uppuluri MV. (2020) Synthesis and biological evaluation of some novel 1,2,3-triazole hybrids of myrrhanone B isolated from Commiphora mukul gum resin: Identification of potent antiproliferative leads active against prostate cancer cells (PC-3)., 188 [PMID:31883489] [10.1016/j.ejmech.2019.111974] |
| 90. Luthra T,Banothu V,Adepally U,Kumar K,M S,Chakrabarti S,Maddi SR,Sen S. (2020) Discovery of novel pyrido-pyrrolidine hybrid compounds as alpha-glucosidase inhibitors and alternative agent for control of type 1 diabetes., 188 [PMID:31927314] [10.1016/j.ejmech.2020.112034] |
| 91. Osella, M. I., Salazar, M. O., Gamarra, M. D., Moreno, D. M., Lambertucci, F., Frances, D. E., Furlan, R. L. E.. (2020) Arylsulfonyl histamine derivatives as powerful and selective alpha-glucosidase inhibitors, 11 (4): [PMID:33479653] [10.1039/c9md00559e] |
| 92. Yu X,Zhang F,Liu T,Liu Z,Dong Q,Li D. (2020) Exploring efficacy of natural-derived acetylphenol scaffold inhibitors for α-glucosidase: Synthesis, in vitro and in vivo biochemical studies., 30 (23): [PMID:32920141] [10.1016/j.bmcl.2020.127528] |
| 93. Duong TH,Paramita Devi A,Tran NM,Phan HV,Huynh NV,Sichaem J,Tran HD,Alam M,Nguyen TP,Nguyen HH,Chavasiri W,Nguyen TC. (2020) Synthesis, α-glucosidase inhibition, and molecular docking studies of novel N-substituted hydrazide derivatives of atranorin as antidiabetic agents., 30 (17): [PMID:32738998] [10.1016/j.bmcl.2020.127359] |
| 94. Bernhard Ellinger, Justus Dick, Vanessa Lage-Rupprecht, Bruce Schultz, Andrea Zaliani, Marcin Namysl, Stephan Gebel, Ole Pless, Jeanette Reinshagen, Christian Ebeling, Alexander Esser, Marc Jacobs, Carsten Claussen, and Martin Hofmann-Apitius. (2021) HDAC6 screening dataset using tau-based substrate in an enzymatic assay yields selective inhibitors and activators, [10.6019/CHEMBL4808148] |
| 95. Chaidam S, Saehlim N, Athipornchai A, Sirion U, Saeeng R.. (2021) Synthesis and biological evaluation of 1,6-bis-triazole-2,3,4-tri-O-benzyl-α-d-glucopyranosides as a novel α-glucosidase inhibitor in the treatment of Type 2 diabetes., 50 [PMID:34418573] [10.1016/j.bmcl.2021.128331] |
| 96. Patel OPS, Jesumoroti OJ, Legoabe LJ, Beteck RM.. (2021) Metronidazole-conjugates: A comprehensive review of recent developments towards synthesis and medicinal perspective., 210 [PMID:33234343] [10.1016/j.ejmech.2020.112994] |
| 97. Li YS, He M, Zhou TS, Wang Q, He L, Wang SJ, Hu B, Wei B, Wang H, Cui ZN.. (2021) 2,5-Disubstituted furan derivatives containing 1,3,4-thiadiazole moiety as potent α-glucosidase and E. coli β-glucuronidase inhibitors., 216 [PMID:33652353] [10.1016/j.ejmech.2021.113322] |
| 98. Umm-E-Farwa, Ullah S, Khan MA, Zafar H, Atia-Tul-Wahab, Younus M, Choudhary MI, Basha FZ.. (2021) Dibenzazepine-linked isoxazoles: New and potent class of α-glucosidase inhibitors., 40 [PMID:33766763] [10.1016/j.bmcl.2021.127979] |
| 99. Gutiérrez-González JA, Pérez-Vásquez A, Torres-Colín R, Rangel-Grimaldo M, Rebollar-Ramos D, Mata R.. (2021) α-Glucosidase Inhibitors from Ageratina grandifolia., 84 (5.0): [PMID:33857371] [10.1021/acs.jnatprod.1c00105] |
| 100. Liang C, Kjaerulff L, Hansen PR, Kongstad KT, Staerk D.. (2021) Dual High-Resolution α-Glucosidase and PTP1B Inhibition Profiling Combined with HPLC-PDA-HRMS-SPE-NMR Analysis for the Identification of Potentially Antidiabetic Chromene Meroterpenoids from Rhododendron capitatum., 84 (9.0): [PMID:34460246] [10.1021/acs.jnatprod.1c00454] |
| 101. Zhang JH, Xie HX, Li Y, Wang KM, Song Z, Zhu KK, Fang L, Zhang J, Jiang CS.. (2021) Design, synthesis and biological evaluation of novel (E)-2-benzylidene-N-(3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)hydrazine-1-carboxamide derivatives as α-glucosidase inhibitors., 52 [PMID:34634473] [10.1016/j.bmcl.2021.128413] |
| 102. Wang SJ, Yu M, Li H, Zhang GJ.. (2022) Structures and Biological Activities of Polyacylated ent-Kaurane Diterpenoid Glycosides from the Aerial Parts of Inula hupehensis., 85 (1.0): [PMID:34964626] [10.1021/acs.jnatprod.1c00947] |
| 103. Huang SZ, Wang Q, Yuan JZ, Cai CH, Wang H, Mándi A, Kurtán T, Dai HF, Zhao YX.. (2022) Hexahydroazulene-2(1H)-one Sesquiterpenoids with Bridged Cyclobutane, Oxetane, and Tetrahydrofuran Rings from the Stems of Daphne papyracea with α-Glycosidase Inhibitory Activity., 85 (1.0): [PMID:34935371] [10.1021/acs.jnatprod.0c01394] |
| 104. Matada BS, Pattanashettar R, Yernale NG.. (2021) A comprehensive review on the biological interest of quinoline and its derivatives., 32 [PMID:33444846] [10.1016/j.bmc.2020.115973] |
| 105. Jiang X, Wu K, Bai R, Zhang P, Zhang Y.. (2022) Functionalized quinoxalinones as privileged structures with broad-ranging pharmacological activities., 229 [PMID:34998058] [10.1016/j.ejmech.2021.114085] |
| 106. Wu Y, Liu C, Hu L.. (2022) Fragment-Based Dynamic Combinatorial Chemistry for Identification of Selective α-Glucosidase Inhibitors., 13 (11.0): [PMID:36385930] [10.1021/acsmedchemlett.2c00405] |
| 107. Le TK, Danova A, Aree T, Duong TH, Koketsu M, Ninomiya M, Sawada Y, Kamsri P, Pungpo P, Chavasiri W.. (2022) α-Glucosidase Inhibitors from the Stems of Knema globularia., 85 (4.0): [PMID:35262352] [10.1021/acs.jnatprod.1c00765] |
| 108. Maurya AK, Baliyan N, Kumar R, Agnihotri VK.. (2022) Synthesis of Sulfur-Containing Analogues of Hedychenone, a Labdane Diterpenoid from Hedychium spicatum., 85 (7.0): [PMID:35790346] [10.1021/acs.jnatprod.2c00112] |
| 109. Simone MI, Wood A, Campkin D, Kiefel MJ, Houston TA.. (2022) Recent results from non-basic glycosidase inhibitors: How structural diversity can inform general strategies for improving inhibition potency., 235 [PMID:35367706] [10.1016/j.ejmech.2022.114282] |
| 110. Oulous A, Daoudi NE, Harit T, Cherfi M, Bnouham M, Malek F.. (2022) New pyrazole-tetrazole hybrid compounds as potent α-amylase and non-enzymatic glycation inhibitors., 69 [PMID:35569687] [10.1016/j.bmcl.2022.128785] |
| 111. Xu T, Meng JR, Cheng W, Liu JZ, Chu J, Zhang Q, Ma N, Bai LP, Guo Y.. (2022) Discovery of honokiol thioethers containing 1,3,4-oxadiazole moieties as potential α-glucosidase and SARS-CoV-2 entry inhibitors., 67 [PMID:35617790] [10.1016/j.bmc.2022.116838] |
| 112. Wu Y, Zhao S, Hu L.. (2022) Identification of potent α-amylase inhibitors via dynamic combinatorial chemistry., 55 [PMID:35021143] [10.1016/j.bmc.2022.116609] |
| 113. Klochkov VG, Bezsonova EN, Dubar M, Melekhina DD, Temnov VV, Zaryanova EV, Lozinskaya NA, Babkov DA, Spasov AA.. (2022) Towards multi-target antidiabetic agents: In vitro and in vivo evaluation of 3,5-disubstituted indolin-2-one derivatives as novel α-glucosidase inhibitors., 55 [PMID:34780899] [10.1016/j.bmcl.2021.128449] |
| 114. İmamoğlu R, Koç E, Kısa D.. (2022) Polyphenolic compounds: Synthesis, assessment of antimicrobial effect and enzymes inhibition against important medicinal enzymes with computational details., 65 [PMID:35395370] [10.1016/j.bmcl.2022.128722] |
| 115. Zhang X, Xu L, Chen H, Zhang X, Lei Y, Liu W, Xu H, Ma B, Zhu C.. (2022) Novel Hydroxychalcone-Based Dual Inhibitors of Aldose Reductase and α-Glucosidase as Potential Therapeutic Agents against Diabetes Mellitus and Its Complications., 65 (13.0): [PMID:35749671] [10.1021/acs.jmedchem.2c00380] |
| 116. Wang KM, Ge YX, Zhang J, Chen YT, Zhang NY, Gu JS, Fang L, Zhang XL, Zhang J, Jiang CS.. (2023) New cycloalkyl[b]thiophenylnicotinamide-based α-glucosidase inhibitors as promising anti-diabetic agents: Synthesis, in silico study, in vitro and in vivo evaluations., 79 [PMID:36395995] [10.1016/j.bmcl.2022.129069] |
| 117. Haider K, Haider MR, Neha K, Yar MS.. (2020) Free radical scavengers: An overview on heterocyclic advances and medicinal prospects., 204 [PMID:32721784] [10.1016/j.ejmech.2020.112607] |
| 118. An Q, Li C, Chen Y, Deng Y, Yang T, Luo Y.. (2020) Repurposed drug candidates for antituberculosis therapy., 192 [PMID:32126450] [10.1016/j.ejmech.2020.112175] |
| 119. Chu J, Yang R, Cheng W, Cui L, Pan H, Liu J, Guo Y.. (2022) Semisynthesis, biological activities, and mechanism studies of Mannich base analogues of magnolol/honokiol as potential α-glucosidase inhibitors., 75 [PMID:36327695] [10.1016/j.bmc.2022.117070] |
| 120. Zhu Y, Zhao J, Luo L, Gao Y, Bao H, Li P, Zhang H.. (2021) Research progress of indole compounds with potential antidiabetic activity., 223 [PMID:34192642] [10.1016/j.ejmech.2021.113665] |
| 121. Elattar KM, El-Khateeb AY, Hamed SE.. (2022) Insights into the recent progress in the medicinal chemistry of pyranopyrimidine analogs., 13 (5.0): [PMID:35694689] [10.1039/d2md00076h] |
| 122. Santos CMM, Freitas M, Fernandes E.. (2018) A comprehensive review on xanthone derivatives as α-glucosidase inhibitors., 157 [PMID:30282319] [10.1016/j.ejmech.2018.07.073] |
| 123. He L, Su Q, Bai L, Li M, Liu J, Liu X, Zhang C, Jiang Z, He J, Shi J, Huang S, Guo L.. (2020) Recent research progress on natural small molecule bibenzyls and its derivatives in Dendrobium species., 204 [PMID:32711292] [10.1016/j.ejmech.2020.112530] |
| 124. Lu L, Chen J, Tao W, Wang Z, Liu D, Zhou J, Wu X, Sun H, Li W, Tanabe G, Muraoka O, Zhao B, Wu L, Xie W.. (2023) Design and Synthesis of Sulfonium Derivatives: A Novel Class of α-Glucosidase Inhibitors with Potent In Vivo Antihyperglycemic Activities., 66 (5): [PMID:36812150] [10.1021/acs.jmedchem.2c01984] |
| 125. He M, Li YJ, Shao J, Li YS, Cui ZN.. (2023) Synthesis and biological evaluation of 2,5-disubstituted furan derivatives containing 1,3-thiazole moiety as potential α-glucosidase inhibitors., 83 [PMID:36764471] [10.1016/j.bmcl.2023.129173] |
| 126. Moghadam Farid S, Iraji A, Mojtabavi S, Ghasemi M, Faramarzi MA, Mahdavi M, Barazandeh Tehrani M, Akbarzadeh T, Saeedi M.. (2023) Quinazolinone-1,2,3-triazole-acetamide conjugates as potent α-glucosidase inhibitors: synthesis, enzyme inhibition, kinetic analysis, and molecular docking study., 14 (3): [PMID:36970140] [10.1039/d2md00297c] |
| 127. Chahal S, Punia J, Rani P, Singh R, Mayank, Kumar P, Kataria R, Joshi G, Sindhu J.. (2023) Development of thiazole-appended novel hydrazones as a new class of α-amylase inhibitors with anticancer assets: an in silico and in vitro approach., 14 (4): [PMID:37122544] [10.1039/d2md00431c] |
| 128. Liang C, Ndi C, Kjaerulff L, Semple S, Buirchell B, Coriani S, Møller BL, Staerk D.. (2023) Characterization of Serrulatane Diterpenoids in Eremophila phyllopoda subsp. phyllopoda by Triple High-Resolution α-Glucosidase/PTP1B/Radical Scavenging Profiling, NMR Spectroscopy, DFT-GIAO NMR, and Electronic Circular Dichroism Calculations., 86 (4): [PMID:36880726] [10.1021/acs.jnatprod.2c00692] |
| 129. Han Jeong G, Cho JH, Park KI, Kim K, Hoon Kim T.. (2023) Enzymatic transformation of esculetin as a potent class of α-glucosidase inhibitors., 88 [PMID:37088219] [10.1016/j.bmcl.2023.129302] |
| 130. Faisal M, Saeed A, Shahzad D, Fattah TA, Lal B, Channar PA, Mahar J, Saeed S, Mahesar PA, Larik FA.. (2017) Enzyme inhibitory activities an insight into the structure-Activity relationship of biscoumarin derivatives., 141 [PMID:29032032] [10.1016/j.ejmech.2017.10.009] |
| 131. Zhang HZ, Zhao ZL, Zhou CH.. (2018) Recent advance in oxazole-based medicinal chemistry., 144 [PMID:29288945] [10.1016/j.ejmech.2017.12.044] |
