Deltarasin - 96%, high purity , CAS No.1440898-61-2

Item Number

D125721

Grouped product items
SKU	Size	Availability	Price
D125721-5mg	5mg	In stock	$147.90
D125721-10mg	10mg	In stock	$236.90
D125721-25mg	25mg	In stock	$533.90
D125721-50mg	50mg	In stock	$759.90
D125721-100mg	100mg	In stock	$1,214.90

Basic Description

Specifications & Purity	≥96%
Biochemical and Physiological Mechanisms	Description: IC50 Value: 41±12 nM (binding to PDEδ in cell) [1] Deltarasin is a novel and small molecule inhibitor which can inhibit the KRAS-PDEδ interaction and impairs oncogenic KRAS signalling. Interfering with b
Storage Temp	Store at -20°C
Shipped In	Ice chest + Ice pads
Product Description	Product introduction Deltarasin is an inhibitor of KRAS-PDEδ interaction with Kd of 38 nM for binding to purified PDEδ.

Associated Targets

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Names and Identifiers

IUPAC Name	1-benzyl-2-[4-[(2S)-2-(2-phenylbenzimidazol-1-yl)-2-piperidin-4-ylethoxy]phenyl]benzimidazole
INCHI	InChI=1S/C40H37N5O/c1-3-11-29(12-4-1)27-44-36-17-9-7-15-34(36)42-39(44)32-19-21-33(22-20-32)46-28-38(30-23-25-41-26-24-30)45-37-18-10-8-16-35(37)43-40(45)31-13-5-2-6-14-31/h1-22,30,38,41H,23-28H2/t38-/m1/s1
InChi Key	LTZKEDSUXKTTTC-KXQOOQHDSA-N
Canonical SMILES	C1CNCCC1C(COC2=CC=C(C=C2)C3=NC4=CC=CC=C4N3CC5=CC=CC=C5)N6C7=CC=CC=C7N=C6C8=CC=CC=C8
Isomeric SMILES	C1CNCCC1[C@@H](COC2=CC=C(C=C2)C3=NC4=CC=CC=C4N3CC5=CC=CC=C5)N6C7=CC=CC=C7N=C6C8=CC=CC=C8
Alternate CAS	1440898-82-7
PubChem CID	73292904
Molecular Weight	603.75

Certificates

Enter Lot Number to search for COA:

To view the certificate results,please click on a Lot number.For Lot numbers from past orders,please use our order status section

10 results found

Lot Number	Certificate Type	Date	Item
K2309373	Certificate of Analysis	Oct 10, 2023	D125721
K2309375	Certificate of Analysis	Oct 10, 2023	D125721
K2309376	Certificate of Analysis	Oct 10, 2023	D125721
K2309377	Certificate of Analysis	Oct 10, 2023	D125721
K2309378	Certificate of Analysis	Oct 10, 2023	D125721
K2309379	Certificate of Analysis	Oct 10, 2023	D125721
K2309380	Certificate of Analysis	Oct 10, 2023	D125721
K2309381	Certificate of Analysis	Oct 10, 2023	D125721
K2309409	Certificate of Analysis	Oct 10, 2023	D125721
K2309419	Certificate of Analysis	Oct 10, 2023	D125721

Solution Calculators

Determine the necessary mass, volume, or concentration for preparing a solution.

Determine the dilution needed to prepare a stock solution.

Basic Description