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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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SKU | Size | Availability | Price | Qty |
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D288728-5mg | 5mg | In stock | $83.90 | |
D288728-10mg | 10mg | In stock | $129.90 | |
D288728-25mg | 25mg | In stock | $290.90 | |
D288728-50mg | 50mg | In stock | $528.90 | |
D288728-100mg | 100mg | In stock | $950.90 | |
D288728-200mg | 200mg | In stock | $1,711.90 |
ACh release enhancer
Synonyms | 160588-45-4 | DMP 543 | DMP-543 | XR-543 | 10,10-BIS[(2-FLUORO-4-PYRIDINYL)METHYL]-9(10H)-ANTHRACENONE | 10,10-Bis((2-fluoropyridin-4-yl)methyl)anthracen-9(10H)-one | CHEMBL343822 | DYD4418J7V | DP-543 | 10,10-Bis((2-fluoro-4-pyridyl)methyl)anthrone | 10,10-bis(2-fluoro-4-py |
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Specifications & Purity | ≥98% |
Biochemical and Physiological Mechanisms | Acetylcholine release stimulator. Potently enhances K+-stimulated [3H]-ACh release from rat hippocampal slices (EC50= 700 nM), and increases release of dopamine and glutamate (EC50values are 0.25 and 0.22μM, respectively). Orally activein vivo; increases |
Storage Temp | Store at 2-8°C |
Shipped In | Wet ice |
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Pubchem Sid | 488196401 |
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Pubchem Sid Url | https://pubchem.ncbi.nlm.nih.gov/substance/488196401 |
IUPAC Name | 10,10-bis[(2-fluoropyridin-4-yl)methyl]anthracen-9-one |
INCHI | InChI=1S/C26H18F2N2O/c27-23-13-17(9-11-29-23)15-26(16-18-10-12-30-24(28)14-18)21-7-3-1-5-19(21)25(31)20-6-2-4-8-22(20)26/h1-14H,15-16H2 |
InChi Key | MUJBUUDUXGDXLW-UHFFFAOYSA-N |
Canonical SMILES | C1=CC=C2C(=C1)C(=O)C3=CC=CC=C3C2(CC4=CC(=NC=C4)F)CC5=CC(=NC=C5)F |
Isomeric SMILES | C1=CC=C2C(=C1)C(=O)C3=CC=CC=C3C2(CC4=CC(=NC=C4)F)CC5=CC(=NC=C5)F |
PubChem CID | 9887884 |
Molecular Weight | 412.44 |
Enter Lot Number to search for COA:
To view the certificate results,please click on a Lot number.For Lot numbers from past orders,please use our order status section
Lot Number | Certificate Type | Date | Item |
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C2321722 | Certificate of Analysis | Mar 09, 2023 | D288728 |
C2321741 | Certificate of Analysis | Mar 09, 2023 | D288728 |
C2321748 | Certificate of Analysis | Mar 09, 2023 | D288728 |
C2321754 | Certificate of Analysis | Mar 09, 2023 | D288728 |
C2321755 | Certificate of Analysis | Mar 09, 2023 | D288728 |
C2321758 | Certificate of Analysis | Mar 09, 2023 | D288728 |
C2321760 | Certificate of Analysis | Mar 09, 2023 | D288728 |
C2321761 | Certificate of Analysis | Mar 09, 2023 | D288728 |
C2321768 | Certificate of Analysis | Mar 09, 2023 | D288728 |
C2321775 | Certificate of Analysis | Mar 09, 2023 | D288728 |
C2321778 | Certificate of Analysis | Mar 09, 2023 | D288728 |
C2321789 | Certificate of Analysis | Mar 09, 2023 | D288728 |
Solubility | Solvent:DMSO, Max Conc. mg/mL: 41.24, Max Conc. mM: 100; Solvent:ethanol, Max Conc. mg/mL: 20.62, Max Conc. mM: 50 |
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