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draflazine , CAS No.120770-34-5, Inhibitor of Equilibrative nucleoside transporter 1

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draflazine , CAS No.120770-34-5, Inhibitor of Equilibrative nucleoside transporter 1

Moligand™

CAS#: 120770-34-5
PubChem CID: 60849

Item Number

D609970

Grouped product items
SKU	Size	Availability	Price	Qty
D609970-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,400.90
D609970-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,000.90

View related series

Equilibrative nucleoside transporter 1 Inhibitor

Basic Description

Synonyms	AKOS040741670 \| SCHEMBL215826 \| UNII-0Y25DT968Y \| 2-(AMINOCARBONYL)-N-(4-AMINO-2,6-DICHLOROPHENYL)-4-(5,5-BIS(4-FLUOROPHENYL)PENTYL)-1-PIPERAZINEACETAMIDE \| HY-106841 \| R 75231 \| R75231 \| R-75231 \| Draflazinum [INN-Latin] \| 1-Piperazineacetamide, 2-(amino
Specifications & Purity	Moligand™
Grade	Moligand™
Action Type	INHIBITOR
Mechanism of action	Inhibitor of Equilibrative nucleoside transporter 1

Associated Targets(Human)

SLC29A1 Tclin Equilibrative nucleoside transporter 1 (1 Activities)

Discover Target: SLC29A1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

SLC29A1 Tclin Equilibrative nucleoside transporter 1 (1711 Activities)

Discover Target: SLC29A1

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Associated Targets(non-human)

SARS-CoV-2 (38078 Activities)

Explore this target

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Mechanisms of Action

Mechanism of Action	Action Type	target ID	Target Name	Target Type	Target Organism	Binding Site Name	References

Names and Identifiers

IUPAC Name	1-{[(4-amino-2,6-dichlorophenyl)carbamoyl]methyl}-4-[5,5-bis(4-fluorophenyl)pentyl]piperazine-2-carboxamide
INCHI	InChI=1S/C30H33Cl2F2N5O2/c31-25-15-23(35)16-26(32)29(25)37-28(40)18-39-14-13-38(17-27(39)30(36)41)12-2-1-3-24(19-4-8-21(33)9-5-19)20-6-10-22(34)11-7-20/h4-11,15-16,24,27H,1-3,12-14,17-18,35H2,(H2,36,41)(H,37,40)
InChi Key	IWMYIWLIESDFRZ-UHFFFAOYSA-N
Canonical SMILES	O=C(Nc1c(Cl)cc(cc1Cl)N)CN1CCN(CC1C(=O)N)CCCCC(c1ccc(cc1)F)c1ccc(cc1)F
Isomeric SMILES	C1CN(C(CN1CCCCC(C2=CC=C(C=C2)F)C3=CC=C(C=C3)F)C(=O)N)CC(=O)NC4=C(C=C(C=C4Cl)N)Cl
PubChem CID	60849

Database links

PubChem CID	60849
CAS Registry No.	120770-34-5
ChEMBL Ligand	CHEMBL1628717

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