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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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SKU | Size | Availability | Price | Qty |
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D126355-10mg | 10mg | Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience! | $98.90 | |
D126355-50mg | 50mg | Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience! | $345.90 | |
D126355-250mg | 250mg | In stock | $1,557.90 |
Agonist selective for estrogen-related receptors ERRβ and ERRγ
Synonyms | DY131|95167-41-2|Benzoic acid, p-hydroxy-, (p-(diethylamino)benzylidene)hydrazide|DY 131|GSK 9089|GSK-9089|5VWV92039E|C18H21N3O2|(E)-DY131|Benzoic acid, 4-hydroxy-, ((4-(diethylamino)phenyl)methylene)hydrazide|Benzoic acid, 4-hydroxy-, 2-((4-(diethylamino |
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Specifications & Purity | ≥98% |
Storage Temp | Store at 2-8°C |
Shipped In | Wet ice |
Grade | Moligand™ |
Action Type | AGONIST |
Mechanism of action | Agonist of Estrogen-related receptor-β;Agonist of Estrogen-related receptor-γ |
Product Description | DY131(GSK 9089) is a novel selective agonist of ERRβ and ERRγ; displays minimal activity at ERRα, ERα and ERβ at concentrations up to 30 μM. |
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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IUPAC Name | N-[(E)-[4-(diethylamino)phenyl]methylideneamino]-4-hydroxybenzamide |
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INCHI | InChI=1S/C18H21N3O2/c1-3-21(4-2)16-9-5-14(6-10-16)13-19-20-18(23)15-7-11-17(22)12-8-15/h5-13,22H,3-4H2,1-2H3,(H,20,23)/b19-13+ |
InChi Key | WLKOCYWYAWBGKY-CPNJWEJPSA-N |
Canonical SMILES | CCN(CC)C1=CC=C(C=C1)C=NNC(=O)C2=CC=C(C=C2)O |
Isomeric SMILES | CCN(CC)C1=CC=C(C=C1)/C=N/NC(=O)C2=CC=C(C=C2)O |
PubChem CID | 5497124 |
Molecular Weight | 311.38 |
PubChem CID | 5497124 |
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ChEMBL Ligand | CHEMBL192509 |
BindingDB Ligand | 22439 |
CAS Registry No. | 95167-41-2 |
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Lot Number | Certificate Type | Date | Item |
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D1727042 | Certificate of Analysis | Nov 16, 2022 | D126355 |
Solubility | Solvent:ethanol, Max Conc. mg/mL: 3.11, Max Conc. mM: 10; Solvent:DMSO, Max Conc. mg/mL: 31.14, Max Conc. mM: 100 |
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Refractive Index | 1.57 |
Pictogram(s) | GHS07 |
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Signal | Warning |
Hazard Statements | H315:Causes skin irritation H319:Causes serious eye irritation H335:May cause respiratory irritation |
Precautionary Statements | P261:Avoid breathing dust/fume/gas/mist/vapors/spray. P305+P351+P338:IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses if present and easy to do - continue rinsing. P280:Wear protective gloves/protective clothing/eye protection/face protection. P302+P352:IF ON SKIN: wash with plenty of water. P321:Specific treatment (see ... on this label). P405:Store locked up. P501:Dispose of contents/container to ... P264:Wash hands [and …] thoroughly after handling. P271:Use only outdoors or in a well-ventilated area. P304+P340:IF INHALED: Remove person to fresh air and keep comfortable for breathing. P403+P233:Store in a well-ventilated place. Keep container tightly closed. P362+P364:Take off contaminated clothing and wash it before reuse. P264+P265:Wash hands [and …] thoroughly after handling. Do not touch eyes. P337+P317:If eye irritation persists: Get medical help. P332+P317:If skin irritation occurs: Get medical help. P319:Get medical help if you feel unwell. |