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dysiherbaine , CAS No.185245-55-0, Agonist of GluK1;Agonist of GluK2;Agonist of GluK3;Agonist of GluK4;Agonist of GluK5

Moligand™

CAS#: 185245-55-0
PubChem CID: 9839436

Item Number

D610035

Grouped product items
SKU	Size	Availability	Price	Qty
D610035-1mg	1mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,000.90
D610035-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$4,000.90

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GluK1 Agonist GluK2 Agonist GluK3 Agonist GluK4 Agonist GluK5 Agonist

Grade

Moligand™

Action Type

AGONIST

Mechanism of action

Agonist of GluK1;Agonist of GluK2;Agonist of GluK3;Agonist of GluK4;Agonist of GluK5

Associated Targets

GRIK4 Tclin Glutamate receptor ionotropic, kainate 4 0 Activities

Discover Target: GRIK4

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

GRIK5 Tclin Glutamate receptor ionotropic, kainate 5 0 Activities

Discover Target: GRIK5

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

GRIK1 Tclin Glutamate receptor ionotropic, kainate 1 2 Activities

Discover Target: GRIK1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

GRIK2 Tclin Glutamate receptor ionotropic, kainate 2 2 Activities

Discover Target: GRIK2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

GRIK3 Tclin Glutamate receptor ionotropic, kainate 3 0 Activities

Discover Target: GRIK3

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Names and Identifiers

IUPAC Name	(2R,3aR,6S,7R,7aR)-2-[(2S)-2-amino-2-carboxyethyl]-6-hydroxy-7-(methylamino)-hexahydro-2H-furo[3,2-b]pyran-2-carboxylic acid
INCHI	InChI=1S/C12H20N2O7/c1-14-8-6(15)4-20-7-3-12(11(18)19,21-9(7)8)2-5(13)10(16)17/h5-9,14-15H,2-4,13H2,1H3,(H,16,17)(H,18,19)/t5-,6+,7+,8+,9-,12+/m0/s1
InChi Key	YUSZFKPLFIQTGF-FDNSHYBFSA-N
Canonical SMILES	CN[C@@H]1[C@H](O)CO[C@H]2[C@@H]1O[C@@](C2)(C[C@@H](C(=O)O)N)C(=O)O
Isomeric SMILES	CN[C@@H]1[C@@H](CO[C@H]2[C@@H]1O[C@@](C2)(C[C@@H](C(=O)O)N)C(=O)O)O
PubChem CID	9839436

PubChem CID

CAS Registry No.

ChEMBL Ligand

RCSB PDB Ligand

References

1. Sakai R, Swanson GT, Shimamoto K, Green T, Contractor A, Ghetti A, Tamura-Horikawa Y, Oiwa C, Kamiya H. (2001) Pharmacological properties of the potent epileptogenic amino acid dysiherbaine, a novel glutamate receptor agonist isolated from the marine sponge Dysidea herbacea.. J Pharmacol Exp Ther, 296 (2): (650-8). [PMID:11160654]

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dysiherbaine , CAS No.185245-55-0, Agonist of GluK1;Agonist of GluK2;Agonist of GluK3;Agonist of GluK4;Agonist of GluK5

Basic Description

Associated Targets

GRIK4 Tclin Glutamate receptor ionotropic, kainate 4 0 Activities

GRIK5 Tclin Glutamate receptor ionotropic, kainate 5 0 Activities

GRIK1 Tclin Glutamate receptor ionotropic, kainate 1 2 Activities

GRIK2 Tclin Glutamate receptor ionotropic, kainate 2 2 Activities

GRIK3 Tclin Glutamate receptor ionotropic, kainate 3 0 Activities

Names and Identifiers

Database links

Certificates

Certificate of Analysis(COA)

Related Documents

References

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