Grouped product items

SKU

Size

Availability

Price

Qty

E610084-5mg

5mg

Available within 8-12 weeks(?)

$600.90

E610084-25mg

25mg

Available within 8-12 weeks(?)

$2,000.90

Basic Description

Synonyms	EHT-1864;EHT1864
Specifications & Purity	Moligand™
Grade	Moligand™

Associated Targets(Human)

5637 (630 Activities)

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A 172 (535 Activities)

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A204 (242 Activities)

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A2058 (690 Activities)

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A-375 (9258 Activities)

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A-427 (643 Activities)

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A498 (42825 Activities)

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A673 (619 Activities)

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ACHN (49357 Activities)

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AGS (1999 Activities)

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BT-20 (503 Activities)

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BT-474 (2113 Activities)

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BXPC-3 (2997 Activities)

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CAKI-1 (44928 Activities)

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Calu-3 (339 Activities)

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Calu-6 (398 Activities)

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CAPAN-1 (772 Activities)

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CFPAC-1 (421 Activities)

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COR-L23 (253 Activities)

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Daoy (570 Activities)

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DMS-273 (14108 Activities)

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DU-145 (51482 Activities)

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EVSA-T (142 Activities)

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G-361 (890 Activities)

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G-401 (156 Activities)

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HT-1080 (3966 Activities)

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HT-29 (80576 Activities)

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HuCCT-1 (128 Activities)

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Huh-7 (12904 Activities)

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HuTu80 (255 Activities)

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J82 (505 Activities)

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JAR (316 Activities)

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KM12 (47707 Activities)

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LoVo (4724 Activities)

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M14 (47487 Activities)

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MCF7 (126967 Activities)

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MDA-MB-361 (612 Activities)

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MDA-MB-453 (1139 Activities)

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MES-SA (905 Activities)

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MG-63 (795 Activities)

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NCI-H1975 (4994 Activities)

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MKN-1 (175 Activities)

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MKN-28 (466 Activities)

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MKN-45 (2102 Activities)

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MKN-7 (272 Activities)

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NCI-H358 (882 Activities)

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NCI-N87 (850 Activities)

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NTERA-2-cl-D1 (234 Activities)

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NUGC-3 (976 Activities)

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OVCAR-3 (48710 Activities)

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Associated Targets(non-human)

H4 (48 Activities)

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Names and Identifiers

IUPAC Name	2-(morpholin-4-ylmethyl)-5-[5-[7-(trifluoromethyl)quinolin-4-yl]sulfanylpentoxy]pyran-4-one
INCHI	InChI=1S/C25H27F3N2O4S/c26-25(27,28)18-4-5-20-21(14-18)29-7-6-24(20)35-13-3-1-2-10-33-23-17-34-19(15-22(23)31)16-30-8-11-32-12-9-30/h4-7,14-15,17H,1-3,8-13,16H2
InChi Key	MIDUFIRTIFUTQA-UHFFFAOYSA-N
Canonical SMILES	O=c1cc(occ1OCCCCCSc1ccnc2c1ccc(c2)C(F)(F)F)CN1CCOCC1
Isomeric SMILES	C1COCCN1CC2=CC(=O)C(=CO2)OCCCCCSC3=C4C=CC(=CC4=NC=C3)C(F)(F)F
PubChem CID	9938203

Database links

PubChem CID	9938203
ChEMBL Ligand	CHEMBL1186585

Certificates

Certificate of Analysis(COA)

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References

1. Shutes A, Onesto C, Picard V, Leblond B, Schweighoffer F, Der CJ. (2007) Specificity and mechanism of action of EHT 1864, a novel small molecule inhibitor of Rac family small GTPases.. J Biol Chem, 282 (49): (35666-78). [PMID:17932039]
2. Onesto C, Shutes A, Picard V, Schweighoffer F, Der CJ. (2008) Characterization of EHT 1864, a novel small molecule inhibitor of Rac family small GTPases.. Meth Enzymol, 439 (3): (111-29). [PMID:18374160]

Solution Calculators

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EHT 1864 , CAS No.E610084

Basic Description

Associated Targets(Human)

Associated Targets(non-human)

Names and Identifiers

Database links

Certificates

Certificate of Analysis(COA)

Related Documents

References

Solution Calculators

Molarity Calculator

Dilution Calculator

Reconstitution Calculator

SKU	Size	Availability	Price	Qty
E610084-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$600.90
E610084-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,000.90