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G protein-coupled receptors (GPCRs)
Opioid receptors
ethylketocyclazocine , CAS No.E610209, Agonist of δ receptor;Agonist of κ receptor;Agonist of μ receptor

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ethylketocyclazocine , CAS No.E610209, Agonist of δ receptor;Agonist of κ receptor;Agonist of μ receptor

Moligand™

PubChem CID: 42800

Item Number

E610209

Grouped product items
SKU	Size	Availability	Price	Qty
E610209-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$600.90
E610209-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,000.90

View related series

δ receptor Agonist κ receptor Agonist μ receptor Agonist

Basic Description

Synonyms	10-(Cyclopropylmethyl)-12-ethyl-4-hydroxy-13-methyl-10-azatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-8-one \| GTPL1602 \| 3-(cyclopropylmethyl)-5-ethyl-8-hydroxy-11-methyl-3,4,5,6-tetrahydro-2,6-methano-3-benzazocin-1(2H)-one \| Q27077242 \| (-)-EKC \| 3-Cyclo
Specifications & Purity	Moligand™
Grade	Moligand™
Action Type	AGONIST
Mechanism of action	Agonist of δ receptor;Agonist of κ receptor;Agonist of μ receptor

Associated Targets(Human)

OPRD1 Tclin Delta-type opioid receptor (1 Activities)

Discover Target: OPRD1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

OPRK1 Tclin Kappa-type opioid receptor (1 Activities)

Discover Target: OPRK1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

OPRM1 Tclin Mu-type opioid receptor (1 Activities)

Discover Target: OPRM1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

OPRM1 Tclin Mu opioid receptor (19785 Activities)

Discover Target: OPRM1

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

OPRK1 Tclin Kappa opioid receptor (16155 Activities)

Discover Target: OPRK1

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Associated Targets(non-human)

Sigmar1 Sigma opioid receptor (160 Activities)

Discover Target: Sigmar1

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Mechanisms of Action

Mechanism of Action	Action Type	target ID	Target Name	Target Type	Target Organism	Binding Site Name	References

Names and Identifiers

INCHI	InChI=1S/C19H25NO2/c1-3-13-10-20(9-12-4-5-12)18-11(2)17(13)16-8-14(21)6-7-15(16)19(18)22/h6-8,11-13,17-18,21H,3-5,9-10H2,1-2H3
InChi Key	MOXLMXQSFOOZDO-UHFFFAOYSA-N
Canonical SMILES	CCC1CN(CC2CC2)C2C(C1c1cc(O)ccc1C2=O)C
Isomeric SMILES	CCC1CN(C2C(C1C3=C(C2=O)C=CC(=C3)O)C)CC4CC4
PubChem CID	42800

Database links

PubChem CID	42800
ChEMBL Ligand	CHEMBL71301
BindingDB Ligand	50017232
GPCRdb Ligand	ethylketocyclazocine

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