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Signal Transduction
Metabolism
Amino Acids
Feniralstat - 99%, high purity , CAS No.2166320-76-7

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Feniralstat - 99%, high purity , CAS No.2166320-76-7

≥99%

CAS#: 2166320-76-7
Formula: C₂₆H₂₅F₂N₅O₄
Molecular Weight: 509.50
PubChem CID: 139301832

Item Number

F646248

Grouped product items
SKU	Size	Availability	Price	Qty
F646248-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$544.90
F646248-10mg	10mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$879.90

View related series

Metabolic Enzyme/Protease Ser/Thr Protease

Basic Description

Specifications & Purity	≥99%
Biochemical and Physiological Mechanisms	Feniralstat (compound 30), a pyrazole derivative, is a potent kallikrein inhibitor with an IC 50 of 6.7 nM for Human plasma kallikrein (pKal). Feniralstat has no inhibition on Human KLKl, Human FXIa, Human Factor Xlla (all IC 50 >40 μM).
Storage Temp	Store at -20°C
Shipped In	Ice chest + Ice pads
Product Description	Feniralstat (compound 30), a pyrazole derivative, is a potent kallikrein inhibitor with an IC 50 of 6.7 nM for Human plasma kallikrein (pKal). Feniralstat has no inhibition on Human KLKl, Human FXIa, Human Factor Xlla (all IC 50 >40 μM). Form:Solid

Associated Targets(Human)

F2 Tclin Thrombin (11687 Activities)

Discover Target: F2

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

PLG Tclin Plasminogen (2339 Activities)

Discover Target: PLG

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

KLKB1 Tclin Plasma kallikrein (2047 Activities)

Discover Target: KLKB1

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Associated Targets(non-human)

Trypsin (394 Activities)

Discover Target:

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Kallikrein 1 (28 Activities)

Discover Target:

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Names and Identifiers

Canonical SMILES	COCC1=NN(C=C1C(=O)NCC2=NC=CC(=C2F)OC)CC3=CC=C(C=C3)CN4C=C(C=CC4=O)F
Isomeric SMILES	COCC1=NN(C=C1C(=O)NCC2=NC=CC(=C2F)OC)CC3=CC=C(C=C3)CN4C=C(C=CC4=O)F
PubChem CID	139301832
Molecular Weight	509.50

Certificates

Certificate of Analysis(COA)

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Chemical and Physical Properties

Solubility	DMSO : 100 mg/mL (196.27 mM; ultrasonic and warming and heat to 60°C)

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