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Home Bioactive Small Molecules Grapiprant (CJ-023,423) - 10mM in DMSO, high purity , Prostanoid EP4 receptor antagonist, CAS No.415903-37-6(DMSO), Prostanoid EP4 receptor antagonist
Grapiprant (CJ-023,423) - 10mM in DMSO, high purity , Prostanoid EP4 receptor antagonist, CAS No.415903-37-6(DMSO), Prostanoid EP4 receptor antagonist
Basic Description Synonyms Grapiprant | 415903-37-6 | CJ-023423 | AAT-007 | RQ-00000007 | N-((4-(2-ethyl-4,6-dimethyl-1H-imidazo[4,5-c]pyridin-1-yl)phenethyl)carbamoyl)-4-methylbenzenesulfonamide | CJ 023423 | CJ-023 | CJ-023,423 | RQ-7 | MR-10A7 | UNII-J9F5ZPH7NB | J9F5ZPH7NB | MR10A7 | Grapiprant (CJ-023423 Specifications & Purity Moligand™, 10mM in DMSO Storage Temp Store at -80°C Shipped In Ice chest + Ice pads Grade Moligand™ Action Type ANTAGONIST Mechanism of action Prostanoid EP4 receptor antagonist Product Description Grapiprant (CJ-023,423, AT-001, AAT-007, RQ-00000007, CJ-23423) is a novel selective EP4 Prostaglandin Receptor inhibitor with Ki of 20 nM and 13 nM for rat EP4 receptor and human EP4 receptor, respectively.
Associated Targets(Human) Associated Targets(non-human) Mechanisms of Action Mechanism of Action Action Type target ID Target Name Target Type Target Organism Binding Site Name References
Names and Identifiers IUPAC Name 1-[2-[4-(2-ethyl-4,6-dimethylimidazo[4,5-c]pyridin-1-yl)phenyl]ethyl]-3-(4-methylphenyl)sulfonylurea INCHI InChI=1S/C26H29N5O3S/c1-5-24-29-25-19(4)28-18(3)16-23(25)31(24)21-10-8-20(9-11-21)14-15-27-26(32)30-35(33,34)22-12-6-17(2)7-13-22/h6-13,16H,5,14-15H2,1-4H3,(H2,27,30,32) InChi Key HZVLFTCYCLXTGV-UHFFFAOYSA-N Canonical SMILES CCC1=NC2=C(N1C3=CC=C(C=C3)CCNC(=O)NS(=O)(=O)C4=CC=C(C=C4)C)C=C(N=C2C)C Isomeric SMILES CCC1=NC2=C(N1C3=CC=C(C=C3)CCNC(=O)NS(=O)(=O)C4=CC=C(C=C4)C)C=C(N=C2C)C PubChem CID 11677589 Molecular Weight 491.61
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