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GSK2647544 - 99%, high purity , CAS No.1380426-95-8

≥99%

CAS#: 1380426-95-8
Formula: C₂₄H₁₈ClF₃N₄O₃
Molecular Weight: 502.87
PubChem CID: 57336782

Item Number

G646149

Grouped product items
SKU	Size	Availability	Price	Qty
G646149-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$376.90
G646149-10mg	10mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$670.90

View related series

Metabolic Enzyme/Protease Phospholipase

Basic Description

Specifications & Purity	≥99%
Biochemical and Physiological Mechanisms	GSK2647544 is an orally available, selective inhibitor of Lp-PLA2 . Lipoprotein-associated phospholipase (Lp-PLA2) is a calcium-independent phospholipase A2 with proinflammatory activities that is primarily secreted by monocyte-derived macrophages.
Storage Temp	Protected from light,Store at -80°C
Shipped In	Ice chest + Ice pads
Product Description	GSK2647544 is an orally available, selective inhibitor of Lp-PLA2. Lipoprotein-associated phospholipase (Lp-PLA2) is a calcium-independent phospholipase A2 with proinflammatory activities that is primarily secreted by monocyte-derived macrophages. Form:Solid

Associated Targets(Human)

PLA2G7 Tchem Platelet-activating factor acetylhydrolase (1 Activities)

Discover Target: PLA2G7

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

PLA2G7 Tchem LDL-associated phospholipase A2 (1338 Activities)

Discover Target: PLA2G7

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Liver (3974 Activities)

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Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Associated Targets(non-human)

Rattus norvegicus (775804 Activities)

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Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Pla2g7 Platelet-activating factor acetylhydrolase (22 Activities)

Discover Target: Pla2g7

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Canonical SMILES

C1=CC(=CC=C1CCOC2=NC=C(C(=O)N2)CC3=CN=CN=C3)OC4=CC(=C(C=C4)Cl)C(F)(F)F

Isomeric SMILES

C1=CC(=CC=C1CCOC2=NC=C(C(=O)N2)CC3=CN=CN=C3)OC4=CC(=C(C=C4)Cl)C(F)(F)F

PubChem CID

57336782

Molecular Weight

502.87

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GSK2647544 - 99%, high purity , CAS No.1380426-95-8

Basic Description

Associated Targets(Human)

Associated Targets(non-human)

Names and Identifiers

Certificates

Certificate of Analysis(COA)

Chemical and Physical Properties

Related Documents

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