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GSK5182 - 10mM in DMSO, high purity , CAS No.877387-37-6
Estrogen/progestogen Receptor Agonists
Basic Description Specifications & Purity Moligand™, 10mM in DMSO Biochemical and Physiological Mechanisms GSK5182, 4-hydroxytamoxifen analog, is a specific inverse agonist of estrogen-related receptor γ (ERRγ) that inhibits pro-inflammatory cytokine-induced catabolic factors. Storage Temp Store at -80°C Shipped In Ice chest + Ice pads Grade Moligand™ Product Description Information
GSK5182 GSK5182, 4-hydroxytamoxifen analog, is a specific inverse agonist of estrogen-related receptor γ (ERRγ) that inhibits pro-inflammatory cytokine-induced catabolic factors.
Targets
ERRγ
Product Properties ALogP 5.308 HBD Count 2 Rotatable Bond 10
Associated Targets(Human) Mechanisms of Action Mechanism of Action Action Type target ID Target Name Target Type Target Organism Binding Site Name References
Names and Identifiers IUPAC Name 4-[(Z)-1-[4-[2-(dimethylamino)ethoxy]phenyl]-5-hydroxy-2-phenylpent-1-enyl]phenol INCHI InChI=1S/C27H31NO3/c1-28(2)18-20-31-25-16-12-23(13-17-25)27(22-10-14-24(30)15-11-22)26(9-6-19-29)21-7-4-3-5-8-21/h3-5,7-8,10-17,29-30H,6,9,18-20H2,1-2H3/b27-26- InChi Key ZVSFNBNLNLXEFQ-RQZHXJHFSA-N Canonical SMILES CN(C)CCOC1=CC=C(C=C1)C(=C(CCCO)C2=CC=CC=C2)C3=CC=C(C=C3)O Isomeric SMILES CN(C)CCOC1=CC=C(C=C1)/C(=C(/CCCO)\C2=CC=CC=C2)/C3=CC=C(C=C3)O PubChem CID 6852176 MeSH Entry Terms GSK5182 Molecular Weight 417.54
Chemical and Physical Properties DMSO(mg / mL) Max Solubility 84 DMSO(mM) Max Solubility 201.178330219859 Water(mg / mL) Max Solubility ＜1
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