Idalopirdine is an potent antagonist of the serotonin 6 (5-HT6) receptor. Idalopirdine has been reported to be highly selective over other G-protein coupled receptors. It has K(d) of 0.2nM for the 5-HT6 receptor with 16-fold selectivity over the 5-HT2A
Storage Temp
Store at -20°C
Shipped In
Ice chest + Ice pads
Grade
Moligand™
Action Type
ANTAGONIST
Mechanism of action
Serotonin 6 (5-HT6) receptor antagonist
Product Description
Idalopirdine is a potent, selective 5-HT6 receptor antagonist with a Ki value of 0.83 nM，which can be used in studies of Alzheimer's disease and schizophrenia, among other related disorders.
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