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J 2156 - ≥98%(HPLC), high purity , CAS No.2387505-73-7, Agonist of SST 4 receptor

Moligand™

≥98%(HPLC)

CAS#: 2387505-73-7
Formula: C₂₄H₂₈N₄O₄S.C₂HF₃O₂
Molecular Weight: 582.6
PubChem CID: 11442741

Item Number

J287752

Grouped product items
SKU	Size	Availability	Price	Qty
J287752-10mg	10mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$286.90
J287752-50mg	50mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$909.90

Selective high affinity human sst4agonist

View related series

SST4 receptor Agonist

Basic Description

Synonyms	J-2156 \| 848647-56-3 \| J-2156 TFA salt \| H35JAI9M2X \| (2S)-4-amino-N-[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]-2-[(4-methylnaphthalen-1-yl)sulfonylamino]butanamide \| J 2156 \| (2~{S})-2-[[(2~{S})-4-azanyl-2-[(4-methylnaphthalen-1-yl)sulfonylamino]butanoyl]amino]-3-phen
Specifications & Purity	Moligand™, ≥98%(HPLC)
Biochemical and Physiological Mechanisms	High affinity human somatostatin receptor 4 (sst4) agonist (Ki= 1.2 nM). Displays >400-fold selectivity for human sst4over other human sst receptor subtypes. Exhibits 2 to 3-fold more potent agonismin vitrothan endogenous ligands somatostatin-14 and somat
Storage Temp	Store at -20°C
Shipped In	Ice chest + Ice pads
Grade	Moligand™
Action Type	AGONIST
Mechanism of action	Agonist of SST 4 receptor

Associated Targets(Human)

SSTR4 Tclin Somatostatin receptor type 4 (2 Activities)

Discover Target: SSTR4

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

SSTR2 Tclin Somatostatin receptor 2 (1526 Activities)

Discover Target: SSTR2

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

SSTR4 Tclin Somatostatin receptor 4 (1125 Activities)

Discover Target: SSTR4

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

InChi Key

VTNCZBXJSGKDLS-SFTDATJTSA-N

Canonical SMILES

CC1=CC=C(S(=O)(N[C@H](C(N[C@H](C(N)=O)CC2=CC=CC=C2)=O)CCN)=O)C3=C1C=CC=C3.OC(C(F)(F)F)=O

Isomeric SMILES

CC1=CC=C(C2=CC=CC=C12)S(=O)(=O)N[C@@H](CCN)C(=O)N[C@@H](CC3=CC=CC=C3)C(=O)N

PubChem CID

11442741

Molecular Weight

582.6

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J 2156 - ≥98%(HPLC), high purity , CAS No.2387505-73-7, Agonist of SST 4 receptor

Basic Description

Associated Targets(Human)

Names and Identifiers

Certificates

Certificate of Analysis(COA)

Chemical and Physical Properties

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