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J 2156 - ≥98%(HPLC), high purity , CAS No.2387505-73-7, Agonist of SST 4 receptor
Selective high affinity human sst4agonist
Basic Description Synonyms GTPL10115 | J 2156 | UNII-H35JAI9M2X | (S)-4-Amino-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((4-methylnaphthalene)-1-sulfonamido)butanamide | J2156 | J-2156 | (1'S, 2S)-4-amino-N-(1'-carbamoyl-2'-phenylethyl)-2-(4''-methyl-1''-naphthalenesulfonylamino) Specifications & Purity Moligand™, ≥98%(HPLC) Biochemical and Physiological Mechanisms High affinity human somatostatin receptor 4 (sst4) agonist (Ki= 1.2 nM). Displays >400-fold selectivity for human sst4over other human sst receptor subtypes. Exhibits 2 to 3-fold more potent agonismin vitrothan endogenous ligands somatostatin-14 and somat Storage Temp Store at -20°C Shipped In Ice chest + Ice pads Grade Moligand™ Action Type AGONIST Mechanism of action Agonist of SST 4 receptor
Associated Targets(Human) Mechanisms of Action Mechanism of Action Action Type target ID Target Name Target Type Target Organism Binding Site Name References
Names and Identifiers InChi Key VTNCZBXJSGKDLS-SFTDATJTSA-N Canonical SMILES CC1=CC=C(S(=O)(N[C@H](C(N[C@H](C(N)=O)CC2=CC=CC=C2)=O)CCN)=O)C3=C1C=CC=C3.OC(C(F)(F)F)=O Isomeric SMILES CC1=CC=C(C2=CC=CC=C12)S(=O)(=O)N[C@@H](CCN)C(=O)N[C@@H](CC3=CC=CC=C3)C(=O)N PubChem CID 11442741 Molecular Weight 582.6
Chemical and Physical Properties Solubility Solvent:water, Max Conc. mg/mL: 58.26, Max Conc. mM: 100; Solvent:DMSO, Max Conc. mg/mL: 58.26, Max Conc. mM: 100
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