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KB SRC 4 - ≥98%(HPLC), high purity , CAS No.1380088-03-8

≥98%(HPLC)

CAS#: 1380088-03-8
Formula: C₃₂H₂₃ClN₈
Molecular Weight: 555.03
PubChem CID: 73349077

Item Number

K288228

Grouped product items
SKU	Size	Availability	Price
K288228-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$229.90
K288228-10mg	10mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$283.90
K288228-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$829.90
K288228-50mg	50mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,136.90

Potent and selective c-Src inhibitor

View related series

Protein Tyrosine Kinase/RTK Src Src Kinase Inhibitors

Basic Description

Specifications & Purity	≥98%(HPLC)
Biochemical and Physiological Mechanisms	Potent and selective c-Src inhibitor (Ki= 44 nM); does not inhibit c-Abl at concentrations up to 125μM. Selective between Src family members (Kdvalues are 86, 160, 240, 720, 3200, 4400, and >40,000 nM for c-Src, Lck, Fgr, Yes, Lyn, Hck and Fyn respectivel
Storage Temp	Store at -20°C
Shipped In	Ice chest + Ice pads

Associated Targets(Human)

LCK Tclin Tyrosine-protein kinase LCK (9212 Activities)

Discover Target: LCK

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

YES1 Tclin Tyrosine-protein kinase YES (2781 Activities)

Discover Target: YES1

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

SK-BR-3 (5175 Activities)

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Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

HMEC (560 Activities)

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Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

FGR Tchem Tyrosine-protein kinase FGR (1748 Activities)

Discover Target: FGR

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Associated Targets(non-human)

Hdac6 Histone deacetylase 6 (222 Activities)

Discover Target: Hdac6

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

rep Replicase polyprotein 1ab (378 Activities)

Discover Target: rep

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Names and Identifiers

IUPAC Name	3-(4-chlorophenyl)-1-[3-[3-[(3-phenylphenyl)methyl]triazol-4-yl]phenyl]pyrazolo[3,4-d]pyrimidin-4-amine
INCHI	InChI=1S/C32H23ClN8/c33-26-14-12-23(13-15-26)30-29-31(34)35-20-36-32(29)41(38-30)27-11-5-10-25(17-27)28-18-37-39-40(28)19-21-6-4-9-24(16-21)22-7-2-1-3-8-22/h1-18,20H,19H2,(H2,34,35,36)
InChi Key	UHIZYQVRKSWIFO-UHFFFAOYSA-N
Canonical SMILES	C1=CC=C(C=C1)C2=CC=CC(=C2)CN3C(=CN=N3)C4=CC(=CC=C4)N5C6=NC=NC(=C6C(=N5)C7=CC=C(C=C7)Cl)N
Isomeric SMILES	C1=CC=C(C=C1)C2=CC=CC(=C2)CN3C(=CN=N3)C4=CC(=CC=C4)N5C6=NC=NC(=C6C(=N5)C7=CC=C(C=C7)Cl)N
PubChem CID	73349077
Molecular Weight	555.03

Certificates

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7 results found

Lot Number	Certificate Type	Date	Item
G2415353	Certificate of Analysis	Apr 01, 2024	K288228
G2415354	Certificate of Analysis	Apr 01, 2024	K288228
G2415355	Certificate of Analysis	Apr 01, 2024	K288228
G2415356	Certificate of Analysis	Apr 01, 2024	K288228
G2415357	Certificate of Analysis	Apr 01, 2024	K288228
G2415358	Certificate of Analysis	Apr 01, 2024	K288228
G2415359	Certificate of Analysis	Apr 01, 2024	K288228

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