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Linagliptin - ≥99%, high purity , Dipeptidyl peptidase IV inhibitor, CAS No.668270-12-0, Dipeptidyl peptidase IV inhibitor
Basic Description Synonyms Linagliptin|668270-12-0|Tradjenta|Ondero|BI 1356|BI-1356|Linagliptin (BI-1356)|Trajenta|Trazenta|BI-1356-BS|BS 1356 BS|UNII-3X29ZEJ4R2|3X29ZEJ4R2|CHEBI:68610|BI-1356BS|HSDB 8204|BI 1356 BS|BS-1356-BS|(R)-8-(3-Amino-piperidin-1-yl)-7-but-2-ynyl-3-methyl-1- Specifications & Purity Moligand™, ≥99% Biochemical and Physiological Mechanisms inagliptin is a highly potent, selective CD26 (DPP-4) inhibitor with IC50 of 1 nM. Storage Temp Store at -20°C Shipped In Ice chest + Ice pads Grade Moligand™ Action Type INHIBITOR Mechanism of action Dipeptidyl peptidase IV inhibitor Note 10mg、50mg、100mg卖完停产，不再备货 Product Description Linagliptin is a highly potent, selective DPP-4 inhibitor with IC50 of 1 nM.
Names and Identifiers IUPAC Name 8-[(3R)-3-aminopiperidin-1-yl]-7-but-2-ynyl-3-methyl-1-[(4-methylquinazolin-2-yl)methyl]purine-2,6-dione INCHI InChI=1S/C25H28N8O2/c1-4-5-13-32-21-22(29-24(32)31-12-8-9-17(26)14-31)30(3)25(35)33(23(21)34)15-20-27-16(2)18-10-6-7-11-19(18)28-20/h6-7,10-11,17H,8-9,12-15,26H2,1-3H3/t17-/m1/s1 InChi Key LTXREWYXXSTFRX-QGZVFWFLSA-N Canonical SMILES CC#CCN1C2=C(N=C1N3CCCC(C3)N)N(C(=O)N(C2=O)CC4=NC5=CC=CC=C5C(=N4)C)C Isomeric SMILES CC#CCN1C2=C(N=C1N3CCC[C@H](C3)N)N(C(=O)N(C2=O)CC4=NC5=CC=CC=C5C(=N4)C)C PubChem CID 10096344 Molecular Weight 472.54
Chemical and Physical Properties Solubility Soluble in DMSO (17 mg/ml at 25 °C), water (<1 mg/ml at 25 °C), ethanol (1 mg/ml at 25 °C), 0.5% hyroxyethylcellulose (30 mg/ml at 25 °C), and methanol.
Safety and Hazards(GHS) Pictogram(s) GHS07 Signal Warning Hazard Statements H315: Causes skin irritation
H319: Causes serious eye irritation
H335: May cause respiratory irritation
Precautionary Statements P261: Avoid breathing dust/fume/gas/mist/vapors/spray.
P305+P351+P338: IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses if present and easy to do - continue rinsing.
P280: Wear protective gloves/protective clothing/eye protection/face protection.
P302+P352: IF ON SKIN: wash with plenty of water.
P321: Specific treatment (see ... on this label).
P405: Store locked up.
P501: Dispose of contents/container to ...
P264: Wash hands [and …] thoroughly after handling.
P271: Use only outdoors or in a well-ventilated area.
P304+P340: IF INHALED: Remove person to fresh air and keep comfortable for breathing.
P403+P233: Store in a well-ventilated place. Keep container tightly closed.
P362+P364: Take off contaminated clothing and wash it before reuse.
P264+P265: Wash hands [and …] thoroughly after handling. Do not touch eyes.
P337+P317: If eye irritation persists: Get medical help.
P332+P317: If skin irritation occurs: Get medical help.
P319: Get medical help if you feel unwell.
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