Determine the necessary mass, volume, or concentration for preparing a solution.
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
---|
SKU | Size | Availability | Price | Qty |
---|---|---|---|---|
L413529-5mg | 5mg | Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience! | $88.90 | |
L413529-10mg | 10mg | Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience! | $141.90 | |
L413529-25mg | 25mg | In stock | $284.90 | |
L413529-50mg | 50mg | In stock | $454.90 | |
L413529-100mg | 100mg | In stock | $682.90 |
Casein Kinase Inhibitors
Specifications & Purity | ≥98% |
---|---|
Biochemical and Physiological Mechanisms | Longdaysin is a Casein Kinase inhibitor with IC50 values of 8.8 μM, 5.6 μM, 52 μM and 29 μM for CKIδ, CKIα, ERK2 and CDK7. |
Storage Temp | Protected from light,Store at -20°C |
Shipped In | Ice chest + Ice pads |
Product Description | Information Longdaysin Longdaysin is a Casein Kinase inhibitor with IC50 values of 8.8 μM, 5.6 μM, 52 μM and 29 μM for CKIδ, CKIα, ERK2 and CDK7. Targets CKIα (Cell-free assay); CKIδ (Cell-free assay); CDK7 (Cell-free assay); CDK7 (Cell-free assay); ERK2 (Cell-free assay) 5.6 μM; 8.8 μM; 29 μM; 29 μM; 52 μM |
ALogP | 3.571 |
---|---|
HBD Count | 1 |
Rotatable Bond | 5 |
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
---|
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
---|
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
---|
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
---|
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
---|
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
---|
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
---|
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
---|
IUPAC Name | 9-propan-2-yl-N-[[3-(trifluoromethyl)phenyl]methyl]purin-6-amine |
---|---|
INCHI | InChI=1S/C16H16F3N5/c1-10(2)24-9-23-13-14(21-8-22-15(13)24)20-7-11-4-3-5-12(6-11)16(17,18)19/h3-6,8-10H,7H2,1-2H3,(H,20,21,22) |
InChi Key | REKSFCCYDQMSIN-UHFFFAOYSA-N |
Canonical SMILES | CC(C)N1C=NC2=C(N=CN=C21)NCC3=CC(=CC=C3)C(F)(F)F |
Isomeric SMILES | CC(C)N1C=NC2=C(N=CN=C21)NCC3=CC(=CC=C3)C(F)(F)F |
PubChem CID | 49830252 |
Molecular Weight | 335.33 |
Enter Lot Number to search for COA:
Find and download the COA for your product by matching the lot number on the packaging.
Lot Number | Certificate Type | Date | Item |
---|---|---|---|
F2218309 | Certificate of Analysis | May 30, 2022 | L413529 |
F2218322 | Certificate of Analysis | May 30, 2022 | L413529 |
F2218323 | Certificate of Analysis | May 30, 2022 | L413529 |
F2218324 | Certificate of Analysis | May 30, 2022 | L413529 |
F2218326 | Certificate of Analysis | May 30, 2022 | L413529 |
Solubility | Solubility (25°C) In vitro DMSO: 67 mg/mL (199.8 mM); Ethanol: 67 mg/mL (199.8 mM); Water: Insoluble; |
---|---|
Sensitivity | light sensitive |
DMSO(mg / mL) Max Solubility | 67 |
DMSO(mM) Max Solubility | 199.803178958041 |
Water(mg / mL) Max Solubility | <1 |