Longdaysin - 98%, high purity , CAS No.1353867-91-0

  • ≥98%
Item Number
L413529
Grouped product items
SKUSizeAvailabilityPrice Qty
L413529-5mg
5mg
Available within 4-8 weeks(?)
Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience!
$88.90
L413529-10mg
10mg
Available within 4-8 weeks(?)
Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience!
$141.90
L413529-25mg
25mg
In stock
$284.90
L413529-50mg
50mg
In stock
$454.90
L413529-100mg
100mg
In stock
$682.90

Casein Kinase Inhibitors

Basic Description

Specifications & Purity≥98%
Biochemical and Physiological MechanismsLongdaysin is a Casein Kinase inhibitor with IC50 values of 8.8 μM, 5.6 μM, 52 μM and 29 μM for CKIδ, CKIα, ERK2 and CDK7.
Storage TempProtected from light,Store at -20°C
Shipped InIce chest + Ice pads
Product Description

Information

Longdaysin Longdaysin is a Casein Kinase inhibitor with IC50 values of 8.8 μM, 5.6 μM, 52 μM and 29 μM for CKIδ, CKIα, ERK2 and CDK7.


Targets

CKIα (Cell-free assay); CKIδ (Cell-free assay); CDK7 (Cell-free assay); CDK7 (Cell-free assay); ERK2 (Cell-free assay) 5.6 μM; 8.8 μM; 29 μM; 29 μM; 52 μM

Product Properties

ALogP3.571
HBD Count1
Rotatable Bond5

Associated Targets(Human)

CSNK1D Tchem Casein kinase I delta (4546 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
CDK2 Tchem Cyclin-dependent kinase 2 (9050 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
CSNK1A1 Tchem Casein kinase I alpha (2581 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
MAPK8 Tchem c-Jun N-terminal kinase 1 (5038 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
CCNH Tbio CDK7/Cyclin H/MNAT1 (693 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
CSNK1D Tchem Casein kinase I isoform alpha/delta (40 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID

Associated Targets(non-human)

Mapk1 MAP kinase ERK2 (650 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
Mus musculus (284745 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID

Names and Identifiers

IUPAC Name 9-propan-2-yl-N-[[3-(trifluoromethyl)phenyl]methyl]purin-6-amine
INCHI InChI=1S/C16H16F3N5/c1-10(2)24-9-23-13-14(21-8-22-15(13)24)20-7-11-4-3-5-12(6-11)16(17,18)19/h3-6,8-10H,7H2,1-2H3,(H,20,21,22)
InChi Key REKSFCCYDQMSIN-UHFFFAOYSA-N
Canonical SMILES CC(C)N1C=NC2=C(N=CN=C21)NCC3=CC(=CC=C3)C(F)(F)F
Isomeric SMILES CC(C)N1C=NC2=C(N=CN=C21)NCC3=CC(=CC=C3)C(F)(F)F
PubChem CID 49830252
Molecular Weight 335.33

Certificates

Certificate of Analysis(COA)

Enter Lot Number to search for COA:

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5 results found

Lot NumberCertificate TypeDateItem
F2218309Certificate of AnalysisMay 30, 2022 L413529
F2218322Certificate of AnalysisMay 30, 2022 L413529
F2218323Certificate of AnalysisMay 30, 2022 L413529
F2218324Certificate of AnalysisMay 30, 2022 L413529
F2218326Certificate of AnalysisMay 30, 2022 L413529

Chemical and Physical Properties

SolubilitySolubility (25°C) In vitro DMSO: 67 mg/mL (199.8 mM); Ethanol: 67 mg/mL (199.8 mM); Water: Insoluble;
Sensitivitylight sensitive
DMSO(mg / mL) Max Solubility67
DMSO(mM) Max Solubility199.803178958041
Water(mg / mL) Max Solubility<1

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