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Loxiglumide - ≥97%(HPLC), high purity , CAS No.107097-80-3, Antagonist of CCK 1 receptor

Moligand™

≥97%(HPLC)

CAS#: 107097-80-3
Formula: C₂₁H₃₀Cl₂N₂O₅
Molecular Weight: 461.38
PubChem CID: 60182

Item Number

L288035

Grouped product items
SKU	Size	Availability	Price
L288035-5mg	5mg	In stock	$43.90
L288035-25mg	25mg	In stock	$198.90
L288035-100mg	100mg	Available within 4-8 weeks(?) Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience!	$497.90

CCK1 antagonist; activein vivo

View related series

CCK1 receptor Antagonist Cholecystokinin Receptor GPCR/G Protein Neuronal Signaling

Basic Description

Synonyms	J-523898 \| GTPL892 \| 4-[(3,4-dichlorobenzoyl)amino]-5-(3-methoxypropyl-pentylamino)-5-oxopentanoic acid \| CCG-221884 \| DTXSID6057615 \| Loxiglumide [INN] \| 4-(3,4-dichlorobenzamido)-5-((3-methoxypropyl)(pentyl)amino)-5-oxopentanoic acid \| BL166440 \| A84729
Specifications & Purity	Moligand™, ≥97%(HPLC)
Biochemical and Physiological Mechanisms	CCK1 antagonist. Suppresses CCK-induced proliferation of acinar cells. Inhibits pancreatic secretion of digestive enzymes. Activein vivo.
Storage Temp	Store at -20°C
Shipped In	Ice chest + Ice pads
Grade	Moligand™
Action Type	ANTAGONIST
Mechanism of action	Antagonist of CCK 1 receptor

Associated Targets(Human)

CCKAR Tclin Cholecystokinin receptor type A (1 Activities)

Discover Target: CCKAR

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Homo sapiens (32628 Activities)

Explore this target

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Associated Targets(non-human)

Cckar Cholecystokinin A receptor (90 Activities)

Discover Target: Cckar

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

rep Replicase polyprotein 1ab (378 Activities)

Discover Target: rep

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Names and Identifiers

IUPAC Name	4-[(3,4-dichlorobenzoyl)amino]-5-[3-methoxypropyl(pentyl)amino]-5-oxopentanoic acid
INCHI	InChI=1S/C21H30Cl2N2O5/c1-3-4-5-11-25(12-6-13-30-2)21(29)18(9-10-19(26)27)24-20(28)15-7-8-16(22)17(23)14-15/h7-8,14,18H,3-6,9-13H2,1-2H3,(H,24,28)(H,26,27)
InChi Key	QNQZBKQEIFTHFZ-UHFFFAOYSA-N
Canonical SMILES	CCCCCN(CCCOC)C(=O)C(CCC(=O)O)NC(=O)C1=CC(=C(C=C1)Cl)Cl
Isomeric SMILES	CCCCCN(CCCOC)C(=O)C(CCC(=O)O)NC(=O)C1=CC(=C(C=C1)Cl)Cl
PubChem CID	60182
Molecular Weight	461.38

PubChem CID

ChEMBL Ligand

BindingDB Ligand

CAS Registry No.

DrugCentral Ligand

GPCRdb Ligand

Certificates

Certificate of Analysis(COA)

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3 results found

Lot Number	Certificate Type	Date	Item
J2129901	Certificate of Analysis	Aug 13, 2024	L288035
J2129902	Certificate of Analysis	Aug 13, 2024	L288035
J2129914	Certificate of Analysis	Aug 13, 2024	L288035

Safety and Hazards(GHS)

Pictogram(s)	GHS07
Signal	Warning
Hazard Statements	H302:Harmful if swallowed
Precautionary Statements	P501:Dispose of contents/container to ... P264:Wash hands [and …] thoroughly after handling. P270:Do not eat, drink or smoke when using this product. P330:Rinse mouth. P301+P317:IF SWALLOWED: Get medical help.

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Loxiglumide - ≥97%(HPLC), high purity , CAS No.107097-80-3, Antagonist of CCK 1 receptor

Basic Description

Associated Targets(Human)

Associated Targets(non-human)

Mechanisms of Action

Names and Identifiers

Database links

Certificates

Certificate of Analysis(COA)

Chemical and Physical Properties

Safety and Hazards(GHS)

Related Documents

Solution Calculators

Molarity Calculator

Dilution Calculator

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