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MEDICA 16 - 98%, high purity , CAS No.87272-20-6, Agonist of FFA1 receptor

Moligand™

≥98%

CAS#: 87272-20-6
Formula: C₂₀H₃₈O₄
Molecular Weight: 342.51
PubChem CID: 121871

Item Number

M288258

Grouped product items
SKU	Size	Availability	Price
M288258-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$89.90
M288258-10mg	10mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$139.90
M288258-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$309.90
M288258-50mg	50mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$509.90
M288258-100mg	100mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$819.90

FFA1 (GPR40) agonist; also inhibits ATP citrate lyase

View related series

ATP Citrate Lyase FFA1 receptor Agonist Free Fatty Acid Receptor GPCR/G Protein Metabolic Enzyme/Protease

Basic Description

Synonyms	3,3,14,14-Tetramethyl-hexadecane-1,16-dioic acid \| SR-01000946665 \| di-tert-butyl[2',4',6'-tris(propan-2-yl)-[1,1'-biphenyl]-2-yl]phosphane \| TC257FLPCK \| Q27132978 \| 3,3,14,14-Tetramethylhexadecanedioic acid \| 3,3,14,14-Tetramethyl-hexadecanedioic acid \|
Specifications & Purity	Moligand™, ≥98%
Biochemical and Physiological Mechanisms	Free fatty acid 1 (FFA1/GPR40) receptor agonist; exhibits selectivity for FFA1 (GPR40) over GPR120. Also inhibits ATP citrate lyase; reduces intracellular triacylglycerol levels in muscle, inhibits lipogenesis and increases insulin sensitivity in rodentsi
Storage Temp	Store at -20°C,Argon charged
Shipped In	Ice chest + Ice pads
Grade	Moligand™
Action Type	AGONIST
Mechanism of action	Agonist of FFA1 receptor

Associated Targets(Human)

FFAR1 Tchem Free fatty acid receptor 1 (1 Activities)

Discover Target: FFAR1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

VDR Tclin Vitamin D receptor (26531 Activities)

Discover Target: VDR

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

ACLY Tclin ATP-citrate synthase (168 Activities)

Discover Target: ACLY

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

POLK Tbio DNA polymerase kappa (8653 Activities)

Discover Target: POLK

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

TDP1 Tchem Tyrosyl-DNA phosphodiesterase 1 (345557 Activities)

Discover Target: TDP1

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Associated Targets(non-human)

Hdac6 Histone deacetylase 6 (222 Activities)

Discover Target: Hdac6

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Echs1 Enoyl-CoA hydratase 1 (14 Activities)

Discover Target: Echs1

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Rattus norvegicus (775804 Activities)

Explore this target

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

GCN5 Histone acetyltransferase GCN5 (89 Activities)

Discover Target: GCN5

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

rep Replicase polyprotein 1ab (378 Activities)

Discover Target: rep

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

fba Putative fructose-1,6-bisphosphate aldolase (15559 Activities)

Discover Target: fba

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Names and Identifiers

IUPAC Name	3,3,14,14-tetramethylhexadecanedioic acid
INCHI	InChI=1S/C20H38O4/c1-19(2,15-17(21)22)13-11-9-7-5-6-8-10-12-14-20(3,4)16-18(23)24/h5-16H2,1-4H3,(H,21,22)(H,23,24)
InChi Key	HYSMCRNFENOHJH-UHFFFAOYSA-N
Canonical SMILES	CC(C)(CCCCCCCCCCC(C)(C)CC(=O)O)CC(=O)O
Isomeric SMILES	CC(C)(CCCCCCCCCCC(C)(C)CC(=O)O)CC(=O)O
PubChem CID	121871
Molecular Weight	342.51

PubChem CID

ChEMBL Ligand

BindingDB Ligand

CAS Registry No.

GPCRdb Ligand

Certificates

Certificate of Analysis(COA)

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8 results found

Lot Number	Certificate Type	Date	Item
A2426323	Certificate of Analysis	Dec 25, 2023	M288258
A2426324	Certificate of Analysis	Dec 25, 2023	M288258
A2426325	Certificate of Analysis	Dec 25, 2023	M288258
A2426326	Certificate of Analysis	Dec 25, 2023	M288258
A2426327	Certificate of Analysis	Dec 25, 2023	M288258
A2426328	Certificate of Analysis	Dec 25, 2023	M288258
A2426329	Certificate of Analysis	Dec 25, 2023	M288258
A2426331	Certificate of Analysis	Dec 25, 2023	M288258

Solubility

Solvent:DMSO, Max Conc. mg/mL: 34.25, Max Conc. mM: 100; Solvent:ethanol, Max Conc. mg/mL: 34.25, Max Conc. mM: 100

Sensitivity

Moisture sensitive

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MEDICA 16 - 98%, high purity , CAS No.87272-20-6, Agonist of FFA1 receptor

Basic Description

Associated Targets(Human)

Associated Targets(non-human)

Mechanisms of Action

Names and Identifiers

Database links

Certificates

Certificate of Analysis(COA)

Chemical and Physical Properties

Related Documents

Solution Calculators

Molarity Calculator

Dilution Calculator

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