MM-433593 , CAS No.M611963, Inhibitor of Fatty acid amide hydrolase

Item Number
M611963
Grouped product items
SKUSizeAvailabilityPrice Qty
M611963-5mg
5mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$1,300.90
M611963-25mg
25mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$2,000.90

Basic Description

SynonymsMM-433593 | 1006604-91-6 | CHEMBL4202707 | ET9Q0750O6 | 2-(1-(4-Chlorobenzyl)-2,5-dimethyl-1h-indol-3-yl)-N-(2-methoxypyridin-4-yl)-2-oxoacetamide | 2-[1-[(4-chlorophenyl)methyl]-2,5-dimethylindol-3-yl]-N-(2-methoxypyridin-4-yl)-2-oxoacetamide | 1H-Indole-3-acetamide
Specifications & PurityMoligand™
GradeMoligand™
Action TypeINHIBITOR
Mechanism of actionInhibitor of Fatty acid amide hydrolase

Associated Targets(Human)

FAAH Tchem Fatty-acid amide hydrolase 1 (2 Activities)
Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)
CNR1 Tclin Cannabinoid CB1 receptor (20913 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID

Associated Targets(non-human)

Faah Anandamide amidohydrolase (3907 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
Rhesus monkey (3147 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID

Names and Identifiers

IUPAC Name 2-[1-[(4-chlorophenyl)methyl]-2,5-dimethylindol-3-yl]-N-(2-methoxypyridin-4-yl)-2-oxoacetamide
INCHI InChI=1S/C25H22ClN3O3/c1-15-4-9-21-20(12-15)23(16(2)29(21)14-17-5-7-18(26)8-6-17)24(30)25(31)28-19-10-11-27-22(13-19)32-3/h4-13H,14H2,1-3H3,(H,27,28,31)
InChi Key RIKZRSJVZWKHNX-UHFFFAOYSA-N
Canonical SMILES COc1nccc(c1)NC(=O)C(=O)c1c2cc(C)ccc2n(c1C)Cc1ccc(cc1)Cl
Isomeric SMILES CC1=CC2=C(C=C1)N(C(=C2C(=O)C(=O)NC3=CC(=NC=C3)OC)C)CC4=CC=C(C=C4)Cl
PubChem CID 25143721

Certificates

Certificate of Analysis(COA)

Enter Lot Number to search for COA:

Related Documents

References

1. Banijamali AR, Wakefield JD, Mermerian AH, Busby RW.  (2014)  Metabolism and disposition of MM-433593, a selective FAAH-1 inhibitor, in monkeys..  Pharmacol Res Perspect,  (5): (e00059).  [PMID:25505606]

Solution Calculators