MRS 1754 - ≥98%, high purity , CAS No.264622-58-4, Antagonist of A 1 receptor;Antagonist of A 2A receptor;Antagonist of A 2B receptor;Antagonist of A 3 receptor

Item Number

M275233

• Synonyms: N-(4-cyanophenyl)-2-[4-(2,6-dioxo-1,3-dipropyl-7H-purin-8-yl)phenoxy]acetamide | (4-Cyano-phenyl)-carbamic acid 4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-phenyl ester | AKOS000346342 | HY-14121 | Lopac0_000729 | 7E435V2DAH | AI3-10031 |
• Specifications & Purity: Moligand™, ≥98%
• Biochemical and Physiological Mechanisms: Selective A 2B antagonist (K i values are 1.97 (hA 2B ), 403 (hA 1 ), 503 (hA 2A ), and 570 nM (hA 3 ).MRS 1754 is a p-cyanoanilide xanthine derivative. It might act as a potential anti-asthmatic drug. MRS 1754 is a potent A2B adenosine receptor antagonis
• Storage Temp: Store at -20°C,Desiccated
• Shipped In: Ice chest + Ice pads
• Grade: Moligand™
• Action Type: ANTAGONIST
• Mechanism of action: Antagonist of A 1 receptor;Antagonist of A 2A receptor;Antagonist of A 2B receptor;Antagonist of A 3 receptor
• Note: Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour. Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.

Product Description

MRS 1754 is a selective antagonist radioligand for A2B adenosine receptor with very low affinity for A1 and A3 receptors of both humans and rats。