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Targets
G protein-coupled receptors (GPCRs)
Bradykinin receptors
N-[(1S)-1-[3-chloro-5-fluoro-2-[[2-methyl-4-(2-methyl-1,2,4-triazol-3-yl)quinolin-8-yl]oxymethyl]phenyl]ethyl]-2-(difluoromethoxy)acetamide , CAS No.N609205, Antagonist of B 2 receptor

N-[(1S)-1-[3-chloro-5-fluoro-2-[[2-methyl-4-(2-methyl-1,2,4-triazol-3-yl)quinolin-8-yl]oxymethyl]phenyl]ethyl]-2-(difluoromethoxy)acetamide , CAS No.N609205, Antagonist of B 2 receptor

Item Number

N609205

Grouped product items
SKU	Size	Availability	Price	Qty
N609205-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,334.90
N609205-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,000.90

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Basic Description

BDKRB2 Tclin B2 bradykinin receptor (0 Activities)

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

IUPAC Name	N-[(1S)-1-[3-chloro-5-fluoro-2-[[2-methyl-4-(2-methyl-1,2,4-triazol-3-yl)quinolin-8-yl]oxymethyl]phenyl]ethyl]-2-(difluoromethoxy)acetamide
INCHI	InChI=1S/C25H23ClF3N5O3/c1-13-7-18(24-30-12-31-34(24)3)16-5-4-6-21(23(16)32-13)36-10-19-17(8-15(27)9-20(19)26)14(2)33-22(35)11-37-25(28)29/h4-9,12,14,25H,10-11H2,1-3H3,(H,33,35)/t14-/m0/s1
InChi Key	ZTCLCSCHTACERP-AWEZNQCLSA-N
Canonical SMILES	FC(OCC(=O)N[C@H](c1cc(F)cc(c1COc1cccc2c1nc(C)cc2c1ncnn1C)Cl)C)F
Isomeric SMILES	CC1=CC(=C2C=CC=C(C2=N1)OCC3=C(C=C(C=C3Cl)F)[C@H](C)NC(=O)COC(F)F)C4=NC=NN4C
PubChem CID	138634054

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1. Lesage A, Gibson C, Marceau F, Ambrosi HD, Saupe J, Katzer W, Loenders B, Charest-Morin X, Knolle J. (2020) In Vitro Pharmacological Profile of a New Small Molecule Bradykinin B₂ Receptor Antagonist.. Front Pharmacol, 11 (13): (916). [PMID:32636746] [10.1021/op500134e]

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