Potent endogenous cannabinoid and vanilloid receptor agonist. (K i values are 0.25 and 12 μM for CB 1 and CB 2 , respectively). Potent agonist at TRPV1 (VR1) receptors (EC 50 = ~50 nM). Active in vivo .
Storage Temp
Protected from light,Store at -20°C,Argon charged,Desiccated
Shipped In
Ice chest + Ice pads
Grade
Moligand™
Action Type
CHANNEL BLOCKER
Mechanism of action
Channel blocker of TRPM8;Channel blocker of TRPV1
Note
Providing storage is as stated on the product vial and the vial is kept tightly sealed, the product can be stored for up to 6 months. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour. Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
Product Description
Store at -20°C (desiccating conditions).
Associated Targets(Human)
TRPV1TclinTransient receptor potential cation channel subfamily V member 1 (1 Activities)