Naftopidil - ≥98.0%, high purity , Alpha-1d adrenergic receptor antagonist, CAS No.57149-07-2, Alpha-1d adrenergic receptor antagonist

Item Number

N129805

• Synonyms: naftopidil | 57149-07-2 | Flivas | KT-611 | Naftopidil [INN] | Avishot | 1-(4-(2-methoxyphenyl)piperazin-1-yl)-3-(naphthalen-1-yloxy)propan-2-ol | BM-15275 | R9PHW59SFN | NSC-759293 | 1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-(naphthalen-1-yloxy)propan-2-ol | CHEMBL142635 | DTXSID
• Specifications & Purity: ≥98%
• Biochemical and Physiological Mechanisms: Naftopidil is an α-1-Adrenergic receptor antagonist and an antihypertensive.α 1 Adrenoceptor antagonist. pK i values are 3.7, 20 and 1.2 for α 1a , α 1b and α 1d , respectively. Orally active. Implicated in benign prostate hyperplasia and bladder obstruct
• Storage Temp: Store at -20°C
• Shipped In: Ice chest + Ice pads
• Action Type: ANTAGONIST
• Mechanism of action: Alpha-1d adrenergic receptor antagonist
• Note: Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour. Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.

Product Description

Naftopidil is a selective α1-adrenergic receptor antagonist or alpha blocker with a Ki of 58.3 nM.
N α-1-Adrenergic receptor antagonist and an antihypertensive.