Nefazodone Hydrochloride - 98%, high purity , Norepinephrine transporter inhibitor, CAS No.82752-99-6, Norepinephrine transporter inhibitor

Item Number

N159830

• Synonyms: CAS-82752-99-6 | AC-1373 | KS-1088 | Tox21_113574 | SCHEMBL41119 | 1-(3-(4-(m-Chlorophenyl)-1-piperazinyl)propyl)-3-ethyl-4-(2-phenoxyethyl)-delta(sup 2)-1,2,4-triazolin-5-one monohydrochloride | 2-[3-[4-(3-Chlorophenyl)-1-piperazinyl]propyl]-5-ethyl-2,4-
• Specifications & Purity: ≥98%
• Biochemical and Physiological Mechanisms: Potent 5-HT 2A receptor antagonist (K i = 7.1 nM for inhibition of [ 3 H] ketanserin binding in rat cortex). Additionally blocks α 1 adrenoceptors (K i values are 5.5 and 84 nM at α 1 and α 2 , respectively).
• Shipped In: Normal
• Action Type: INHIBITOR
• Mechanism of action: Norepinephrine transporter inhibitor
• Note: Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour. Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.