Determine the necessary mass, volume, or concentration for preparing a solution.
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
---|
SKU | Size | Availability | Price | Qty |
---|---|---|---|---|
O288423-5mg | 5mg | In stock | $122.90 | |
O288423-10mg | 10mg | In stock | $211.90 | |
O288423-25mg | 25mg | In stock | $477.90 | |
O288423-50mg | 50mg | In stock | $637.90 | |
O288423-100mg | 100mg | In stock | $1,148.90 |
Potent LSD1 inhibitor
Specifications & Purity | Moligand™, ≥98%(HPLC) |
---|---|
Biochemical and Physiological Mechanisms | Potent LSD1 inhibitor (IC50= 20 nM). Exhibits some selectivity for LSD1 over MAO-B and MAO-A (IC50values are 0.72 and 1.38 μM, respectively). Inhibits herpes simplex virus (HSV) immediate early gene expression and viral yieldin vitro. Suppresses HSV prima |
Storage Temp | Store at -20°C |
Shipped In | Ice chest + Ice pads |
Grade | Moligand™ |
Action Type | INHIBITOR |
Mechanism of action | Inhibitor of lysine demethylase 1A |
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
---|
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
---|
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
---|
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
---|
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
---|
Mechanism of Action | Action Type | target ID | Target Name | Target Type | Target Organism | Binding Site Name | References |
---|
IUPAC Name | 3-[4-[(1R,2S)-2-aminocyclopropyl]phenyl]phenol |
---|---|
INCHI | InChI=1S/C15H15NO/c16-15-9-14(15)11-6-4-10(5-7-11)12-2-1-3-13(17)8-12/h1-8,14-15,17H,9,16H2/t14-,15+/m1/s1 |
InChi Key | DSOJSZXQRJGBCW-CABCVRRESA-N |
Canonical SMILES | C1C(C1N)C2=CC=C(C=C2)C3=CC(=CC=C3)O |
Isomeric SMILES | C1[C@@H]([C@H]1N)C2=CC=C(C=C2)C3=CC(=CC=C3)O |
PubChem CID | 56639570 |
Molecular Weight | 225.29 |
PubChem CID | 56639570 |
---|---|
CAS Registry No. | 1357302-64-7 |
Enter Lot Number to search for COA:
Find and download the COA for your product by matching the lot number on the packaging.
Lot Number | Certificate Type | Date | Item |
---|---|---|---|
K2222591 | Certificate of Analysis | Mar 09, 2022 | O288423 |
K2222598 | Certificate of Analysis | Mar 09, 2022 | O288423 |
K2222604 | Certificate of Analysis | Mar 09, 2022 | O288423 |
K2222605 | Certificate of Analysis | Mar 09, 2022 | O288423 |
K2222607 | Certificate of Analysis | Mar 09, 2022 | O288423 |
Solubility | Solvent:DMSO, Max Conc. mg/mL: 22.53, Max Conc. mM: 100; Solvent:ethanol, Max Conc. mg/mL: 22.53, Max Conc. mM: 100; Solvent:1eq. HCl, Max Conc. mg/mL: 4.51, Max Conc. mM: 20 |
---|