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Home Cardiovascular Heart Autophagy OPC 21268 - ≥98%(HPLC), high purity , CAS No.131631-89-5, Antagonist of OT receptor;Antagonist of V 1A receptor;Antagonist of V 2 receptor
OPC 21268 - ≥98%(HPLC), high purity , CAS No.131631-89-5, Antagonist of OT receptor;Antagonist of V 1A receptor;Antagonist of V 2 receptor
Basic Description Synonyms Pharmakon1600-01301020 | 3-(DIMETHYLDODECYLAMMONIO)PROPANE-1-SULFONATE | F0001-0544 | CS-0003694 | FT-0700164 | A856968 | MS-28145 | N-(3-(4-(4-(2-oxo-3,4-dihydroquinolin-1(2H)-yl)piperidine-1-carbonyl)phenoxy)propyl)acetamide | BCP14853 | GTPL2196 | SCHE Specifications & Purity Moligand™, ≥98%(HPLC) Biochemical and Physiological Mechanisms Nonpeptide Vasotocin V1receptor antagonist. Displays greater affinity for rat V1than human V1(Kivalues are 25 and 8800 nM respectively). Exhibits 1000-fold selectivity for V1receptors over V2receptors. Orally active.OPC-21268 is one of 2 non-peptide V1a s Storage Temp Store at -20°C Shipped In Ice chest + Ice pads Grade Moligand™ Action Type ANTAGONIST Mechanism of action Antagonist of OT receptor;Antagonist of V 1A receptor;Antagonist of V 2 receptor Product Description Product description：
Fuscoside (OPC-21268) is an orally effective, nonpeptide, Vasotocin V1 receptor antagonist with an IC50 of 0.4 μM.
Associated Targets(Human) Associated Targets(non-human) Mechanisms of Action Mechanism of Action Action Type target ID Target Name Target Type Target Organism Binding Site Name References
Names and Identifiers Pubchem Sid 488187520 Pubchem Sid Url https://pubchem.ncbi.nlm.nih.gov/substance/488187520 IUPAC Name N-[3-[4-[4-(2-oxo-3,4-dihydroquinolin-1-yl)piperidine-1-carbonyl]phenoxy]propyl]acetamide INCHI InChI=1S/C26H31N3O4/c1-19(30)27-15-4-18-33-23-10-7-21(8-11-23)26(32)28-16-13-22(14-17-28)29-24-6-3-2-5-20(24)9-12-25(29)31/h2-3,5-8,10-11,22H,4,9,12-18H2,1H3,(H,27,30) InChi Key KSNUCNRMDYJBKT-UHFFFAOYSA-N Canonical SMILES CC(=O)NCCCOC1=CC=C(C=C1)C(=O)N2CCC(CC2)N3C(=O)CCC4=CC=CC=C43 Isomeric SMILES CC(=O)NCCCOC1=CC=C(C=C1)C(=O)N2CCC(CC2)N3C(=O)CCC4=CC=CC=C43 PubChem CID 114904 Molecular Weight 449.54
Chemical and Physical Properties Solubility Solvent:DMSO, Max Conc. mg/mL: 44.95, Max Conc. mM: 100; Solvent:ethanol, Max Conc. mg/mL: 11.24, Max Conc. mM: 25
Safety and Hazards(GHS) Pictogram(s) GHS09 , GHS07 Signal Warning Hazard Statements H302: Harmful if swallowed
H400: Very toxic to aquatic life
Precautionary Statements P273: Avoid release to the environment.
P501: Dispose of contents/container to ...
P264: Wash hands [and …] thoroughly after handling.
P270: Do not eat, drink or smoke when using this product.
P391: Collect spillage.
P330: Rinse mouth.
P301+P317: IF SWALLOWED: Get medical help.
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