PBD-150 - 10mM in DMSO, high purity , CAS No.790663-33-1

Item Number
P425969
Grouped product items
SKUSizeAvailabilityPrice Qty
P425969-1ml
1ml
Available within 4-8 weeks(?)
Items will be manufactured post-order and can take 4-8 weeks. Thank you for your patience!
$241.90

Basic Description

Specifications & PurityMoligand™, 10mM in DMSO
Biochemical and Physiological MechanismsPBD-150 is a human\xa0glutaminyl cyclase (hQC) Y115E-Y117E\xa0variant inhibitor with Ki of 490 nM.
Storage TempStore at -80°C
Shipped InIce chest + Ice pads
GradeMoligand™
Product Description

Information

PBD-150 is a human glutaminyl cyclase (hQC) Y115E-Y117E variant inhibitor with Ki of 490 nM.

Associated Targets(Human)

QPCT Tchem Glutaminyl-peptide cyclotransferase (3 Activities)
Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)
QPCT Tchem Glutaminyl-peptide cyclotransferase (1121 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID

Mechanisms of Action

Mechanism of ActionAction Typetarget IDTarget NameTarget TypeTarget OrganismBinding Site NameReferences

Names and Identifiers

IUPAC Name 1-(3,4-dimethoxyphenyl)-3-(3-imidazol-1-ylpropyl)thiourea
INCHI InChI=1S/C15H20N4O2S/c1-20-13-5-4-12(10-14(13)21-2)18-15(22)17-6-3-8-19-9-7-16-11-19/h4-5,7,9-11H,3,6,8H2,1-2H3,(H2,17,18,22)
InChi Key FZQXMGLQANXZRP-UHFFFAOYSA-N
Canonical SMILES COC1=C(C=C(C=C1)NC(=S)NCCCN2C=CN=C2)OC
Isomeric SMILES COC1=C(C=C(C=C1)NC(=S)NCCCN2C=CN=C2)OC
PubChem CID 6539196
Molecular Weight 320.4

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