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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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SKU | Size | Availability | Price | Qty |
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P276048-5mg | 5mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $55.90 | |
P276048-25mg | 25mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $178.90 | |
P276048-50mg | 50mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $284.90 | |
P276048-100mg | 100mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $455.90 |
Cell permeable, selective, non-peptidic calpain inhibitor
Specifications & Purity | ≥95% |
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Biochemical and Physiological Mechanisms | Cell permeable, selective, non-peptidic calpain inhibitor (K i values are 0.3 and 5 μM for calpain 1 and calpain 2, respectively). Stimulates phagocyte function via hFPR/hFPRL1 activation. Interacts with the Ca 2+ calpain sites. |
Storage Temp | Protected from light,Store at -20°C,Desiccated |
Shipped In | Ice chest + Ice pads |
Note | Unstable; make up solutions fresh and use immediately. Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details. |
Product Description | Store at -20°C. Store In the Dark. Store under desiccating conditions. This product is air and light sensitive and impurities can occur as a result of air oxidation or due to metabolism by microbes. |
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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IUPAC Name | (Z)-3-(5-fluoro-1H-indol-3-yl)-2-sulfanylprop-2-enoic acid |
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INCHI | InChI=1S/C11H8FNO2S/c12-7-1-2-9-8(4-7)6(5-13-9)3-10(16)11(14)15/h1-5,13,16H,(H,14,15)/b10-3- |
InChi Key | HWMQHECFXSVZGN-KMKOMSMNSA-N |
Canonical SMILES | C1=CC2=C(C=C1F)C(=CN2)C=C(C(=O)O)S |
Isomeric SMILES | C1=CC2=C(C=C1F)C(=CN2)/C=C(/C(=O)O)\S |
WGK Germany | 3 |
PubChem CID | 5353866 |
Molecular Weight | 237.25 |
Enter Lot Number to search for COA:
Find and download the COA for your product by matching the lot number on the packaging.
Lot Number | Certificate Type | Date | Item |
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G2402290 | Certificate of Analysis | Mar 06, 2024 | P276048 |
G2408173 | Certificate of Analysis | Mar 06, 2024 | P276048 |
G2408174 | Certificate of Analysis | Mar 06, 2024 | P276048 |
G2408225 | Certificate of Analysis | Mar 06, 2024 | P276048 |
G2408230 | Certificate of Analysis | Mar 06, 2024 | P276048 |
G2408231 | Certificate of Analysis | Mar 06, 2024 | P276048 |
G2408232 | Certificate of Analysis | Mar 06, 2024 | P276048 |
G2408234 | Certificate of Analysis | Mar 06, 2024 | P276048 |
Solubility | Soluble in DMSO to 100 mM |
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Sensitivity | air and light sensitive |
WGK Germany | 3 |
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RIDADR | NONHforallmodesoftransport |
Starting at $210.90