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SKU | Size | Availability | Price | Qty |
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P648963-5mg | 5mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $210.90 | |
P648963-10mg | 10mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $330.90 | |
P648963-50mg | 50mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $1,160.90 |
Synonyms | Perzinfotel | 144912-63-0 | EAA-090 | FX5AUU7Z8T | WAY-126090 | (2-(8,9-Dioxo-2,6-diazabicyclo(5.2.0)non-1(7)-en-2-yl)ethyl)phosphonic acid | [2-(8,9-dioxo-2,6-diazabicyclo[5.2.0]non-1(7)-en-2-yl)ethyl]phosphonic acid | Phosphonic acid, (2-(8,9-dioxo-2,6-diazabicyclo(5 |
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Specifications & Purity | ≥98% |
Biochemical and Physiological Mechanisms | Perzinfotel (EAA-090) is a potent, selective, and competitive NMDA receptor antagonist with neuroprotective effects. Perzinfotel (EAA-090) shows high affinity ( IC 50 =30 nM) for the glutamate site. |
Storage Temp | Store at -20°C |
Shipped In | Ice chest + Ice pads |
Action Type | ANTAGONIST |
Mechanism of action | Glutamate [NMDA] receptor antagonist |
Product Description | Perzinfotel (EAA-090) is a potent, selective, and competitive NMDA receptor antagonist with neuroprotective effects. Perzinfotel (EAA-090) shows high affinity ( IC 50 =30 nM) for the glutamate site In Vitro Perzinfotel blocks NMDA-induced currents with an IC 50 of 0.48 μM and glutamate-induced neurotoxicity with an IC 50 of 1.6 μM. MCE has not independently confirmed the accuracy of these methods. They are for reference only. Form:Solid IC50& Target:NMDA receptor |
ALogP | -1.6 |
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IUPAC Name | 2-(8,9-dioxo-2,6-diazabicyclo[5.2.0]non-1(7)-en-2-yl)ethylphosphonic acid |
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INCHI | InChI=1S/C9H13N2O5P/c12-8-6-7(9(8)13)11(3-1-2-10-6)4-5-17(14,15)16/h10H,1-5H2,(H2,14,15,16) |
InChi Key | BDABGOLMYNHHTR-UHFFFAOYSA-N |
Canonical SMILES | C1CNC2=C(C(=O)C2=O)N(C1)CCP(=O)(O)O |
Isomeric SMILES | C1CNC2=C(C(=O)C2=O)N(C1)CCP(=O)(O)O |
WGK Germany | 3 |
PubChem CID | 6918236 |
Molecular Weight | 260.18 |
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Solubility | DMSO : 20.83 mg/mL (80.06 mM; Need ultrasonic) H2O : 5.88 mg/mL (22.60 mM; ultrasonic and warming and heat to 60°C) |
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Pictogram(s) | GHS06 |
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Signal | Danger |
Hazard Statements | H300:Fatal if swallowed |
Precautionary Statements | P321:Specific treatment (see ... on this label). P405:Store locked up. P501:Dispose of contents/container to ... P264:Wash hands [and …] thoroughly after handling. P270:Do not eat, drink or smoke when using this product. P330:Rinse mouth. P301+P316:IF SWALLOWED: Get emergency medical help immediately. |
WGK Germany | 3 |
RIDADR | UN28116.1/PGIII |