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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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SKU | Size | Availability | Price | Qty |
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P287273-10mg | 10mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $499.90 | |
P287273-50mg | 50mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $1,499.90 |
Competitive NMDA antagonist
Synonyms | 113919-36-1|PMPA (NMDA antagonist)|4-(PHOSPHONOMETHYL)PIPERAZINE-2-CARBOXYLIC ACID|2-Piperazinecarboxylic acid, 4-(phosphonomethyl)-|Pmpa(nmda antagonist)|4-(Phosphonomethyl)-2-piperazinecarboxylic acid|CHEMBL29244|SCHEMBL1999794|DTXSID30590848|AKOS024457 |
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Biochemical and Physiological Mechanisms | Competitive NMDA receptor antagonist. Displays Kivalues of 0.84, 2.74, 3.53 and 4.16μM at GluN2A, GluN2B, GluN2C and GluN2D subunit-containing receptors respectively. Selective over AMPA receptors.Please refer toIUPHAR Guide to Pharmacologyfor the most re |
Storage Temp | Store at 2-8°C |
Shipped In | Wet ice |
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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IUPAC Name | 4-(phosphonomethyl)piperazine-2-carboxylic acid |
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INCHI | InChI=1S/C6H13N2O5P/c9-6(10)5-3-8(2-1-7-5)4-14(11,12)13/h5,7H,1-4H2,(H,9,10)(H2,11,12,13) |
InChi Key | ILRBBHJXTYIHTP-UHFFFAOYSA-N |
Canonical SMILES | C1CN(CC(N1)C(=O)O)CP(=O)(O)O |
Isomeric SMILES | C1CN(CC(N1)C(=O)O)CP(=O)(O)O |
PubChem CID | 17756792 |
Molecular Weight | 224.15 |
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Solubility | Solvent:water, Max Conc. mg/mL: 22.42, Max Conc. mM: 100 |
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