PP121 - ≥98%, high purity , CAS No.1092788-83-4, Inhibitor of ABL proto-oncogene 1; non-receptor tyrosine kinase;Inhibitor of epidermal growth factor receptor;Inhibitor of HCK proto-oncogene; Src family tyrosine kinase;Inhibitor of kinase insert domain receptor;Inhibitor of mechanistic target of rapamyc
PP121 - ≥98%, high purity , CAS No.1092788-83-4, Inhibitor of ABL proto-oncogene 1; non-receptor tyrosine kinase;Inhibitor of epidermal growth factor receptor;Inhibitor of HCK proto-oncogene; Src family tyrosine kinase;Inhibitor of kinase insert domain receptor;Inhibitor of mechanistic target of rapamyc
Inhibitor of ABL proto-oncogene 1; non-receptor tyrosine kinase;Inhibitor of epidermal growth factor receptor;Inhibitor of HCK proto-oncogene; Src family tyrosine kinase;Inhibitor of kinase insert domain receptor;Inhibitor of mechanistic target of rapamyc
Product Description
PP-121 is a multi-targeted inhibitor of PDGFR, Hck, mTOR, VEGFR2, Src and Abl with IC50 of 2 nM, 8 nM, 10 nM, 12 nM, 14 nM and 18 nM, also inhibits DNA-PK with IC50 of 60 nM. An inhibitor of c-Abl, PI 3-kinase, PDGFR, Hck, FRAP, Flk-1, SRC, and DNA-PK.