Determine the necessary mass, volume, or concentration for preparing a solution.
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SKU | Size | Availability | Price | Qty |
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P288242-5mg | 5mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $117.90 | |
P288242-10mg | 10mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $197.90 | |
P288242-25mg | 25mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $385.90 | |
P288242-50mg | 50mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $593.90 | |
P288242-100mg | 100mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $890.90 |
High affinity and selective P2Y14antagonist
Specifications & Purity | ≥98%(HPLC) |
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Biochemical and Physiological Mechanisms | High affinity and selective P2Y14antagonist (KB= 434 pM). Exhibits >10,000-fold selectivity for P2Y14over other P2Y receptors. Inhibits UDP-glucose andMRS 2690-induced porcine pancreatic artery contractionex vivo. Also blocks UDP-glucose-induced chemotaxi |
Storage Temp | Store at -20°C |
Shipped In | Ice chest + Ice pads |
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IUPAC Name | 4-(4-piperidin-4-ylphenyl)-7-[4-(trifluoromethyl)phenyl]naphthalene-2-carboxylic acid;hydrochloride |
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INCHI | InChI=1S/C29H24F3NO2.ClH/c30-29(31,32)25-8-5-19(6-9-25)22-7-10-26-23(15-22)16-24(28(34)35)17-27(26)21-3-1-18(2-4-21)20-11-13-33-14-12-20;/h1-10,15-17,20,33H,11-14H2,(H,34,35);1H |
InChi Key | FKMVYPCBLWYNAV-UHFFFAOYSA-N |
Canonical SMILES | C1CNCCC1C2=CC=C(C=C2)C3=C4C=CC(=CC4=CC(=C3)C(=O)O)C5=CC=C(C=C5)C(F)(F)F.Cl |
Isomeric SMILES | C1CNCCC1C2=CC=C(C=C2)C3=C4C=CC(=CC4=CC(=C3)C(=O)O)C5=CC=C(C=C5)C(F)(F)F.Cl |
PubChem CID | 121513852 |
Molecular Weight | 512 |
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Solubility | Solvent:DMSO, Max Conc. mg/mL: 51.2, Max Conc. mM: 100; Solvent:ethanol, Max Conc. mg/mL: 10.24, Max Conc. mM: 20 |
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