PROTAC ERRα ligand 2 - 10mM in DMSO, high purity , CAS No.2306388-57-6(DMSO)

  • 10mM in DMSO
Item Number
P655477
Grouped product items
SKUSizeAvailabilityPrice Qty
P655477-1ml
1ml
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$198.90

Basic Description

Specifications & Purity10mM in DMSO
Biochemical and Physiological MechanismsPROTAC ERRα ligand 2 is an estrogen-related receptor α ( ERRα ) inverse agonist with an IC 50 of 5.67 nM. PROTAC ERRα ligand 2 (IC 50 =5.67 nM) displays a ~11-fold improved potency than XCT790 (IC 50 =61.3 nM).
Storage TempStore at -80°C
Shipped InIce chest + Ice pads
Product Description

PROTAC ERRα ligand 2 is an estrogen-related receptor α ( ERRα ) inverse agonist with an IC 50 of 5.67 nM. PROTAC ERRα ligand 2 (IC 50 =5.67 nM) displays a ~11-fold improved potency than XCT790 (IC 50 =61.3 nM).

Associated Targets(Human)

ESRRA Tchem Steroid hormone receptor ERR1 (1 Activities)
Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

Names and Identifiers

Canonical SMILES COC1=C(C=CC(=C1)C=C(C#N)C(=O)O)OCC2=C(C=C(C=C2)C(F)(F)F)C(F)(F)F
Molecular Weight 445.3

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