Proteasome Inhibitor VII, Antiprotealide - ≥95%, high purity , CAS No.11173422

  • ≥95%
Item Number
P390560
Grouped product items
SKUSizeAvailabilityPrice Qty
P390560-50μg
50μg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$379.90

Basic Description

Specifications & Purity≥95%
Storage TempStore at -80°C
Shipped InIce chest + Ice pads
Product Description

Proteasome Inhibitor VII, Antiprotealide is a cell-permeable, Omuralide-Salinosporamide hybrid that irreversibly inactivates the β5-subunit of the human 20S proteasome. The compound has shown to be ~2.5-fold more potent than Omuralide and is expected to exhibit comparable whole cell potency to Salinosporamide A.
Proteasome Inhibitor VII, Antiprotealideis which inactivates the β5-subunit of the human 20S proteasome

Product Properties

pKapKₐ: 13.27 (Predicted)

Associated Targets(Human)

RPMI-8226 (44974 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID
HCT-116 (91556 Activities)
Activity TypeRelationActivity valueUnitsAction TypeJournalPubMed IddoiAssay Aladdin ID

Names and Identifiers

Canonical SMILES CC(C)[C@@H]([C@H]12C(=O)O[C@H]1([C@H](C(=O)N2)CCCl)C)O
Isomeric SMILES CC(C)[C@@H]([C@]12C(=O)O[C@]1([C@H](C(=O)N2)CCCl)C)O
PubChem CID 11173422
Molecular Weight 275.7

Certificates

Certificate of Analysis(COA)

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Chemical and Physical Properties

SolubilitySoluble in DMSO.
Refractive Indexn20D1.53 (Predicted)
Boil Point(°C)484.69° C at 760 mmHg (Predicted)
Melt Point(°C)194.33° C (Predicted)

Related Documents

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