Determine the necessary mass, volume, or concentration for preparing a solution.
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
---|
SKU | Size | Availability | Price | Qty |
---|---|---|---|---|
R129875-50mg | 50mg | In stock | $58.90 | |
R129875-250mg | 250mg | In stock | $265.90 | |
R129875-1g | 1g | In stock | $955.90 | |
R129875-5g | 5g | In stock | $4,301.90 |
MAO-B inhibitor
Synonyms | (1R)-2,3-Dihydro-N-2-propynyl-1H-in den-1-amine methanesulfonate | s2102 | D02562 | MFCD08460604 | 1H-INDEN-1-AMINE, 2,3-DIHYDRO-N-2-PROPYNYL-, (R)-, METHANESULPHONATE | Rasagiline mesylate [USAN] | 1H-Inden-1-amine, 2,3-dihydro-N-2-propyn-1-yl-, (1R)-, m |
---|---|
Specifications & Purity | ≥99% |
Biochemical and Physiological Mechanisms | Rasagiline Mesylate is an antiparkinsonian and a selective irreversible MAO-B inhibitor. Rasagiline mesylate is an effective therapeutic option in early stages of Parkinson′s disease. It improves the motor fluctuations in levodopa-treated patients and may |
Storage Temp | Store at 2-8°C |
Shipped In | Wet ice |
Action Type | INHIBITOR |
Mechanism of action | Monoamine oxidase B inhibitor |
Note | Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour. Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details. |
Product Description | Rasagiline Mesylate is a new MAO-B inhibitor for the treatment of idiopathic Parkinson's disease. |
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
---|
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
---|
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
---|
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
---|
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
---|
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
---|
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
---|
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
---|
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
---|
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
---|
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
---|
Mechanism of Action | Action Type | target ID | Target Name | Target Type | Target Organism | Binding Site Name | References |
---|
IUPAC Name | methanesulfonic acid;(1R)-N-prop-2-ynyl-2,3-dihydro-1H-inden-1-amine |
---|---|
INCHI | InChI=1S/C12H13N.CH4O3S/c1-2-9-13-12-8-7-10-5-3-4-6-11(10)12;1-5(2,3)4/h1,3-6,12-13H,7-9H2;1H3,(H,2,3,4)/t12-;/m1./s1 |
InChi Key | JDBJJCWRXSVHOQ-UTONKHPSSA-N |
Canonical SMILES | CS(=O)(=O)O.C#CCNC1CCC2=CC=CC=C12 |
Isomeric SMILES | CS(=O)(=O)O.C#CCN[C@@H]1CCC2=CC=CC=C12 |
WGK Germany | 3 |
PubChem CID | 3052775 |
Molecular Weight | 267.34 |
Enter Lot Number to search for COA:
Find and download the COA for your product by matching the lot number on the packaging.
Lot Number | Certificate Type | Date | Item |
---|---|---|---|
B23171125 | Certificate of Analysis | Feb 23, 2023 | R129875 |
B23171133 | Certificate of Analysis | Feb 23, 2023 | R129875 |
B23171154 | Certificate of Analysis | Feb 23, 2023 | R129875 |
B2318010 | Certificate of Analysis | Feb 23, 2023 | R129875 |
B2318055 | Certificate of Analysis | Feb 23, 2023 | R129875 |
D1527038 | Certificate of Analysis | Jan 09, 2023 | R129875 |
Solubility | DMSO 53 mg/mL Water 53 mg/mL Ethanol 53 mg/mL |
---|---|
Sensitivity | Heat Sensitive |
Specific Rotation[α] | 21° (C=2,EtOH) |
Melt Point(°C) | 157 °C |
Pictogram(s) | GHS07 |
---|---|
Signal | Warning |
Hazard Statements | H302:Harmful if swallowed |
Precautionary Statements | P501:Dispose of contents/container to ... P264:Wash hands [and …] thoroughly after handling. P270:Do not eat, drink or smoke when using this product. P330:Rinse mouth. P301+P317:IF SWALLOWED: Get medical help. |
WGK Germany | 3 |
Merck Index | 8116 |