Reldesemtiv - ≥97%, high purity , Fast skeletal troponin complex activator, CAS No.1345410-31-2, Fast skeletal troponin complex activator

Item Number

R669809

Grouped product items
SKU	Size	Availability	Price
R669809-1mg	1mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$179.90
R669809-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$389.90
R669809-10mg	10mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$579.90
R669809-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$939.90
R669809-100mg	100mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,760.90
R669809-250mg	250mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$2,934.90

Basic Description

Synonyms	1-(2-(((TRANS-3-FLUORO-1-(3-FLUORO-2-PYRIDINYL)CYCLOBUTYL)METHYL)AMINO)-5-PYRIMIDINYL)- 1H-PYRROLE-3-CARBOXAMIDE \| SCHEMBL12288022 \| 1-[2-[[3-fluoro-1-(3-fluoropyridin-2-yl)cyclobutyl]methylamino]pyrimidin-5-yl]pyrrole-3-carboxamide \| CK-2127107
Specifications & Purity	≥97%
Storage Temp	Store at -20°C
Shipped In	Ice chest + Ice pads
Action Type	ACTIVATOR
Mechanism of action	Fast skeletal troponin complex activator
Product Description	Reldesemtiv is a selective and next-generation fast skeletal muscle troponin activator (FSTA). Reldesemtiv selectively activates fast skeletal myofibrils with an EC50 of 3.4 μM. Reldesemtiv increases exercise performance in a heart failure model.

Associated Targets(Human)

KCNH2 Tclin HERG (29587 Activities)

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

NR1I2 Tchem Pregnane X receptor (6667 Activities)

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Names and Identifiers

IUPAC Name	1-[2-[[3-fluoro-1-(3-fluoropyridin-2-yl)cyclobutyl]methylamino]pyrimidin-5-yl]pyrrole-3-carboxamide
INCHI	InChI=1S/C19H18F2N6O/c20-13-6-19(7-13,16-15(21)2-1-4-23-16)11-26-18-24-8-14(9-25-18)27-5-3-12(10-27)17(22)28/h1-5,8-10,13H,6-7,11H2,(H2,22,28)(H,24,25,26)
InChi Key	MQXWPWOCXGARRK-UHFFFAOYSA-N
Canonical SMILES	NC(=O)C1=CN(C=C1)C2=CN=C(N=C2)NC[C@]3(C[C@@H](F)C3)C4=C(F)C=CC=N4
Isomeric SMILES	C1C(CC1(CNC2=NC=C(C=N2)N3C=CC(=C3)C(=O)N)C4=C(C=CC=N4)F)F
PubChem CID	67454400
Molecular Weight	384.4

Certificates

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5 results found

Lot Number	Certificate Type	Date	Item
H2419158	Certificate of Analysis	May 07, 2024	R669809
H2419159	Certificate of Analysis	May 07, 2024	R669809
H2419160	Certificate of Analysis	May 07, 2024	R669809
H2419161	Certificate of Analysis	May 07, 2024	R669809
H2419162	Certificate of Analysis	May 07, 2024	R669809

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Basic Description