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Regulators of G protein Signaling (RGS) proteins
RGS4 inhibitor 11b , CAS No.410074-60-1, Inhibitor of regulator of G-protein signaling 4;Inhibitor of regulator of G-protein signaling 8

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RGS4 inhibitor 11b , CAS No.410074-60-1, Inhibitor of regulator of G-protein signaling 4;Inhibitor of regulator of G-protein signaling 8

Moligand™

CAS#: 410074-60-1
PubChem CID: 6539137

Item Number

R613174

Grouped product items
SKU	Size	Availability	Price	Qty
R613174-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$271.90
R613174-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$946.90

View related series

regulator of G-protein signaling 4 Inhibitor regulator of G-protein signaling 8 Inhibitor

Basic Description

Synonyms	thiadiazolidinone (TDZD) deriv. 6
Specifications & Purity	Moligand™
Grade	Moligand™
Action Type	INHIBITOR
Mechanism of action	Inhibitor of regulator of G-protein signaling 4;Inhibitor of regulator of G-protein signaling 8

Associated Targets

RGS8 Tchem Regulator of G-protein signaling 8 1 Activities

Discover Target: RGS8

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

RGS4 Tchem Regulator of G-protein signaling 4 2 Activities

Discover Target: RGS4

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

CHRM3 Tclin Muscarinic acetylcholine receptor M3 0 Activities

Discover Target: CHRM3

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

GSK3B Tclin Glycogen synthase kinase-3 beta 0 Activities

Discover Target: GSK3B

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Names and Identifiers

IUPAC Name	4-butyl-2-ethyl-1,2,4-thiadiazolidine-3,5-dione
INCHI	InChI=1S/C8H14N2O2S/c1-3-5-6-9-7(11)10(4-2)13-8(9)12/h3-6H2,1-2H3
InChi Key	WTFFYZGCISALRI-UHFFFAOYSA-N
Canonical SMILES	CCCCn1c(=O)sn(c1=O)CC
Isomeric SMILES	CCCCN1C(=O)N(SC1=O)CC
PubChem CID	6539137

Database links

PubChem CID	6539137
ChEMBL Ligand	CHEMBL24773
CAS Registry No.	410074-60-1

Certificates

Certificate of Analysis(COA)

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References

1. Turner EM, Blazer LL, Neubig RR, Husbands SM. (2012) Small Molecule Inhibitors of Regulator of G Protein Signalling (RGS) Proteins.. ACS Med Chem Lett, 3 (2): (146-150). [PMID:22368763]

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