Determine the necessary mass, volume, or concentration for preparing a solution.
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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SKU | Size | Availability | Price | Qty |
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R613288-5mg | 5mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $1,334.90 | |
R613288-25mg | 25mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $2,000.90 |
Synonyms | RPR-121154 |
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Specifications & Purity | Moligand™ |
Grade | Moligand™ |
Action Type | ANTAGONIST |
Mechanism of action | Antagonist of C5a 1 receptor |
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) |
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Mechanism of Action | Action Type | target ID | Target Name | Target Type | Target Organism | Binding Site Name | References |
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C5a anaphylatoxin chemotactic receptor antagonist | ANTAGONIST | ALA2373 | C5a anaphylatoxin chemotactic receptor | SINGLE PROTEIN | Homo sapiens | PubMed: [1] | |
C5a anaphylatoxin chemotactic receptor inhibitor | INHIBITOR | ALA2373 | C5a anaphylatoxin chemotactic receptor | SINGLE PROTEIN | Homo sapiens |
IUPAC Name | 2-methyl-1-[3-phenyl-4-(2-phenylethoxy)phenyl]guanidine |
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INCHI | InChI=1S/C22H23N3O/c1-24-22(23)25-19-12-13-21(20(16-19)18-10-6-3-7-11-18)26-15-14-17-8-4-2-5-9-17/h2-13,16H,14-15H2,1H3,(H3,23,24,25) |
InChi Key | QXDMVRPQHNFBSZ-UHFFFAOYSA-N |
Canonical SMILES | CN=C(Nc1ccc(c(c1)c1ccccc1)OCCc1ccccc1)N |
Isomeric SMILES | CN=C(N)NC1=CC(=C(C=C1)OCCC2=CC=CC=C2)C3=CC=CC=C3 |
PubChem CID | 10020451 |