RPR121154 , CAS No.R613288, Antagonist of C5a 1 receptor

Item Number
R613288
Grouped product items
SKUSizeAvailabilityPrice Qty
R613288-5mg
5mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$1,334.90
R613288-25mg
25mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$2,000.90

Basic Description

SynonymsRPR-121154
Specifications & PurityMoligand™
GradeMoligand™
Action TypeANTAGONIST
Mechanism of actionAntagonist of C5a 1 receptor

Associated Targets(Human)

C5AR1 Tclin C5a anaphylatoxin chemotactic receptor 1 (1 Activities)
Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)

Mechanisms of Action

Mechanism of ActionAction Typetarget IDTarget NameTarget TypeTarget OrganismBinding Site NameReferences
C5a anaphylatoxin chemotactic receptor antagonistANTAGONISTALA2373C5a anaphylatoxin chemotactic receptorSINGLE PROTEINHomo sapiens

PubMed: [1]


C5a anaphylatoxin chemotactic receptor inhibitorINHIBITORALA2373C5a anaphylatoxin chemotactic receptorSINGLE PROTEINHomo sapiens

Other: [1] , [2]


Names and Identifiers

IUPAC Name 2-methyl-1-[3-phenyl-4-(2-phenylethoxy)phenyl]guanidine
INCHI InChI=1S/C22H23N3O/c1-24-22(23)25-19-12-13-21(20(16-19)18-10-6-3-7-11-18)26-15-14-17-8-4-2-5-9-17/h2-13,16H,14-15H2,1H3,(H3,23,24,25)
InChi Key QXDMVRPQHNFBSZ-UHFFFAOYSA-N
Canonical SMILES CN=C(Nc1ccc(c(c1)c1ccccc1)OCCc1ccccc1)N
Isomeric SMILES CN=C(N)NC1=CC(=C(C=C1)OCCC2=CC=CC=C2)C3=CC=CC=C3
PubChem CID 10020451

Certificates

C of A & Other Certificates

Related Documents

Solution Calculators