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RS 102221 hydrochloride , CAS No.185376-97-0, Antagonist of 5-HT 2A receptor;Antagonist of 5-HT 2B receptor;Antagonist of 5-HT 2C receptor
a selective SR-2C antagonist
Basic Description
| Synonyms | N-[5-[5-(2,4-Dioxo-1,3,8-triazaspiro[4.5]decan-8-yl)-1-oxopentyl]-2,4-dimethoxyphenyl]-4-(trifluoromethyl)benzenesulfonamide | BPBio1_000243 | N-[5-[5-(2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl)pentanoyl]-2,4-dimethoxyphenyl]-4-(trifluoromethyl)benzenesu |
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| Specifications & Purity | Moligand™ |
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| Storage Temp | Store at 2-8°C |
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| Shipped In | Wet ice |
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| Grade | Moligand™ |
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| Action Type | ANTAGONIST |
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| Mechanism of action | Antagonist of 5-HT 2A receptor;Antagonist of 5-HT 2B receptor;Antagonist of 5-HT 2C receptor |
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Associated Targets(Human)
Associated Targets(non-human)
Names and Identifiers
| IUPAC Name | N-[5-[5-(2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl)pentanoyl]-2,4-dimethoxyphenyl]-4-(trifluoromethyl)benzenesulfonamide |
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| INCHI | InChI=1S/C27H31F3N4O7S/c1-40-22-16-23(41-2)20(33-42(38,39)18-8-6-17(7-9-18)27(28,29)30)15-19(22)21(35)5-3-4-12-34-13-10-26(11-14-34)24(36)31-25(37)32-26/h6-9,15-16,33H,3-5,10-14H2,1-2H3,(H2,31,32,36,37) |
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| InChi Key | HZZZZODVDSHQRG-UHFFFAOYSA-N |
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| Canonical SMILES | COC1=CC(=C(C=C1C(=O)CCCCN2CCC3(CC2)C(=O)NC(=O)N3)NS(=O)(=O)C4=CC=C(C=C4)C(F)(F)F)OC |
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| Isomeric SMILES | COC1=CC(=C(C=C1C(=O)CCCCN2CCC3(CC2)C(=O)NC(=O)N3)NS(=O)(=O)C4=CC=C(C=C4)C(F)(F)F)OC |
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| WGK Germany | 3 |
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| Alternate CAS | 185376-97-0 |
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| PubChem CID | 3693566 |
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| MeSH Entry Terms | 8-(5-(5-amino-2,4-dimethoxyphenyl)-5-oxopentyl)-1,3,8-triazaspiro(4.5)decane-2,4-dione;RS 102221;RS-102221 |
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| Molecular Weight | 649.08 |
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Chemical and Physical Properties
| Solubility | Soluble in DMSO (≥ 20 mg/ml). |
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