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S 38093 - ≥98%(HPLC), high purity , CAS No.1403835-45-9

Item Number

S287735

Grouped product items
SKU	Size	Availability	Price	Qty
S287735-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$68.90
S287735-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$264.90

Selective H3antagonist and inverse agonist; also σ1receptor antagonist; antinociceptive

Basic Description

Synonyms	rel-4-[3-[(3aR,6aS)-Hexahydrocyclopenta[c]pyrrol-2(1H)-yl]propoxy]benzamide
Specifications & Purity	≥98%(HPLC)
Biochemical and Physiological Mechanisms	H3antagonist and inverse agonist (Kivalues are 8.8, 1.2 and 1.44 μM, at rat, human and mouse, respectively). Exhibits no activity at other histaminergic receptors. Antagonizes agonist action at mouse H3receptors (KB= 0.65 μM). Displays inverse agonist act
Storage Temp	Store at -20°C
Shipped In	Ice chest + Ice pads

HRH1 Tclin Histamine H1 receptor (7573 Activities)

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

HRH3 Tclin Histamine H3 receptor (10389 Activities)

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Rattus norvegicus (775804 Activities)

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

IUPAC Name	4-[3-[(3aS,6aR)-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-2-yl]propoxy]benzamide
INCHI	InChI=1S/C17H24N2O2/c18-17(20)13-5-7-16(8-6-13)21-10-2-9-19-11-14-3-1-4-15(14)12-19/h5-8,14-15H,1-4,9-12H2,(H2,18,20)/t14-,15+
InChi Key	MRNMYWNBLVJWKG-GASCZTMLSA-N
Canonical SMILES	C1CC2CN(CC2C1)CCCOC3=CC=C(C=C3)C(=O)N
Isomeric SMILES	C1C[C@@H]2CN(C[C@@H]2C1)CCCOC3=CC=C(C=C3)C(=O)N
PubChem CID	70941112
Molecular Weight	288.39

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Solubility	Solvent:DMSO, Max Conc. mg/mL: 28.84, Max Conc. mM: 100; Solvent:ethanol, Max Conc. mg/mL: 14.42, Max Conc. mM: 50

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