S-(+)-CBPG , CAS No.180465-02-5, Antagonist of mGlu 1 receptor;Agonist of mGlu 5 receptor

Item Number

S386556

Grouped product items
SKU	Size	Availability	Price	Qty
S386556-1mg	1mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$33.90
S386556-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$126.90

a structurally new group I mGluR antagonist

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Basic Description

Specifications & Purity	Moligand™
Storage Temp	Store at 2-8°C
Shipped In	Wet ice
Grade	Moligand™
Action Type	AGONIST, ANTAGONIST
Mechanism of action	Antagonist of mGlu 1 receptor;Agonist of mGlu 5 receptor
Product Description	S-(+)-CBPG is a potent and selective, structurally new group I metabotropic glutamate receptor (mGluR) antagonist. S-(+)-CBPGis a structurally new group I mGluR antagonist

Associated Targets(Human)

GRM1 Tchem Metabotropic glutamate receptor 1 (1 Activities)

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

GRM5 Tchem Metabotropic glutamate receptor 5 (1 Activities)

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

GRM4 Tchem Metabotropic glutamate receptor 4 (2320 Activities)

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

GRM1 Tchem Metabotropic glutamate receptor 1 (2309 Activities)

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

GRM5 Tchem Metabotropic glutamate receptor 5 (5733 Activities)

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Names and Identifiers

IUPAC Name	3-[(S)-amino(carboxy)methyl]bicyclo[1.1.1]pentane-1-carboxylic acid
INCHI	InChI=1S/C8H11NO4/c9-4(5(10)11)7-1-8(2-7,3-7)6(12)13/h4H,1-3,9H2,(H,10,11)(H,12,13)/t4-,7?,8?/m1/s1
InChi Key	KNSHLWJBSDBBRH-XOJFDHPMSA-N
Canonical SMILES	C1C2(CC1(C2)C(=O)O)C(C(=O)O)N
Isomeric SMILES	C1C2(CC1(C2)C(=O)O)[C@@H](C(=O)O)N
PubChem CID	5311040
MeSH Entry Terms	2-(3'-carboxybicyclo(1.1.1)pentyl)glycine;CBPG compound;UPF 596;UPF-596;UPF596
Molecular Weight	185.18

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Basic Description