Potent κ agonist (K i = 8-19 nM). Psychoactive and antinociceptive in vivo . Reported to be an allosteric modulator of μ opioid receptors.
Storage Temp
Store at -20°C,Desiccated
Shipped In
Ice chest + Ice pads
Grade
Moligand™
Action Type
AGONIST
Mechanism of action
Agonist of κ receptor
Note
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour. Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
Product Description
Product Describtion:
Salvinorin A is a non-nitrogenous κ-opioid selective agonist
1.Pittaluga A et al.. (2013) Effects of the neoclerodane Hardwickiic acid on the presynaptic opioid receptors which modulate noradrenaline and dopamine release in mouse central nervous system.. Neurochem Int, 62 (4):(354-9). [PMID:23357481]
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