Determine the necessary mass, volume, or concentration for preparing a solution.
Activity Type | Relation | Activity value | Units | Action Type | Journal | PubMed Id | doi | Assay Aladdin ID |
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SKU | Size | Availability | Price | Qty |
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S275082-1mg | 1mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $59.90 | |
S275082-5mg | 5mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $179.90 | |
S275082-10mg | 10mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $226.90 | |
S275082-25mg | 25mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $589.90 | |
S275082-50mg | 50mg | Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding. | $950.90 |
Selective h5-HT 1B antagonist
Synonyms | SB-216641 HCl | SB216641 | SB216641HYDROCHLORIDE | SB 216641A | HY-103149 | SB216641 hydrochloride | BCP20784 | N-[3-[2-(dimethylamino)ethoxy]-4-methoxyphenyl]-4-[2-methyl-4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]benzamide;hydrochloride | SB-216641A | DTXS |
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Specifications & Purity | ≥97% |
Biochemical and Physiological Mechanisms | Selective h5-HT 1B receptor antagonist. 25-fold selectivity over h5-HT 1D . Little or no affinity for a range of other receptor subtypes. |
Storage Temp | Store at -20°C |
Shipped In | Ice chest + Ice pads |
Note | Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour. Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details. |
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IUPAC Name | N-[3-[2-(dimethylamino)ethoxy]-4-methoxyphenyl]-4-[2-methyl-4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]benzamide;hydrochloride |
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INCHI | InChI=1S/C28H30N4O4.ClH/c1-18-16-22(27-29-19(2)36-31-27)10-12-24(18)20-6-8-21(9-7-20)28(33)30-23-11-13-25(34-5)26(17-23)35-15-14-32(3)4;/h6-13,16-17H,14-15H2,1-5H3,(H,30,33);1H |
InChi Key | JPBMDMNORXKGHZ-UHFFFAOYSA-N |
Canonical SMILES | CC1=C(C=CC(=C1)C2=NOC(=N2)C)C3=CC=C(C=C3)C(=O)NC4=CC(=C(C=C4)OC)OCCN(C)C.Cl |
Isomeric SMILES | CC1=C(C=CC(=C1)C2=NOC(=N2)C)C3=CC=C(C=C3)C(=O)NC4=CC(=C(C=C4)OC)OCCN(C)C.Cl |
PubChem CID | 10392025 |
Molecular Weight | 523.03 |
Enter Lot Number to search for COA:
Find and download the COA for your product by matching the lot number on the packaging.
Lot Number | Certificate Type | Date | Item |
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H2415407 | Certificate of Analysis | Apr 30, 2024 | S275082 |
H2415408 | Certificate of Analysis | Apr 30, 2024 | S275082 |
H2415409 | Certificate of Analysis | Apr 30, 2024 | S275082 |
H2415410 | Certificate of Analysis | Apr 30, 2024 | S275082 |
H2415411 | Certificate of Analysis | Apr 30, 2024 | S275082 |
H2415412 | Certificate of Analysis | Apr 30, 2024 | S275082 |
H2415413 | Certificate of Analysis | Apr 30, 2024 | S275082 |
H2415414 | Certificate of Analysis | Apr 30, 2024 | S275082 |
H2415415 | Certificate of Analysis | Apr 30, 2024 | S275082 |
H2415416 | Certificate of Analysis | Apr 30, 2024 | S275082 |
Solubility | Soluble in water to 25 mM (with warming) |
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