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Sertaconazole nitrate - ≥98%, high purity , Cytochrome P450 51 inhibitor, CAS No.99592-39-9, Cytochrome P450 51 inhibitor

≥98%

CAS#: 99592-39-9
Formula: C₂₀H₁₅Cl₃N₂OS·HNO₃
Molecular Weight: 500.78
PubChem CID: 200103
PubChem SID: 488188600

Item Number

S129395

Grouped product items
SKU	Size	Availability	Price
S129395-10mg	10mg	In stock	$48.90
S129395-50mg	50mg	In stock	$93.90
S129395-250mg	250mg	In stock	$423.90
S129395-500mg	500mg	Available within 1-2 weeks(?) Item is derived from our semi-finished stock and is processed in 1-2 weeks.	$761.90
S129395-1g	1g	In stock	$1,370.90

Basic Description

Synonyms	Sertaconazole nitrate\|99592-39-9\|Dermofix\|Ertaczo\|Zalain\|Sertaconazole mononitrate\|Dermovit\|Ginedermofix\|FI 7056\|Sertaconazole (nitrate)\|DTXSID2045529\|UNII-1DV05410M5\|FI-7045\|1DV05410M5\|FI-7056\|DTXCID0025529\|99592-39-9 (Nitrate)\|1H-Imidazole, 1-(2-((7-chl
Specifications & Purity	≥98%
Biochemical and Physiological Mechanisms	Sertaconazole interacts with 14-alpha demethylase, a cytochrome P-450 enzyme necessary to convert lanosterol to ergosterol. As ergosterol is an essential component of the fungal cell membrane, inhibition of its synthesis results in increased cellular perm
Storage Temp	Store at -20°C
Shipped In	Ice chest + Ice pads
Action Type	INHIBITOR
Mechanism of action	Cytochrome P450 51 inhibitor
Note	卖完停产，不再备货

Associated Targets

EHMT2 Tchem Histone-lysine N-methyltransferase EHMT2 0 Activities

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GMNN Tbio Geminin 0 Activities

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PTH1R Tclin Parathyroid hormone/parathyroid hormone-related peptide receptor 0 Activities

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HSP90AA1 Tchem Heat shock protein HSP 90-alpha 1 Activities

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KAT2A Tchem Histone acetyltransferase KAT2A 0 Activities

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SMAD3 Tchem Mothers against decapentaplegic homolog 3 0 Activities

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L3MBTL1 Tchem Lethal(3)malignant brain tumor-like protein 1 0 Activities

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BAZ2B Tchem Bromodomain adjacent to zinc finger domain protein 2B 0 Activities

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ATXN2 Tbio Ataxin-2 0 Activities

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TDP1 Tchem Tyrosyl-DNA phosphodiesterase 1 0 Activities

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ATAD5 Tbio ATPase family AAA domain-containing protein 5 0 Activities

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GLP1R Tclin Glucagon-like peptide 1 receptor 0 Activities

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IDH1 Tclin Isocitrate dehydrogenase [NADP] cytoplasmic 0 Activities

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NFE2L2 Tchem Nuclear factor erythroid 2-related factor 2 0 Activities

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KDM4A Tchem Lysine-specific demethylase 4A 0 Activities

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Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Names and Identifiers

Pubchem Sid	488188600
Pubchem Sid Url	https://pubchem.ncbi.nlm.nih.gov/substance/488188600
IUPAC Name	1-[2-[(7-chloro-1-benzothiophen-3-yl)methoxy]-2-(2,4-dichlorophenyl)ethyl]imidazole;nitric acid
INCHI	InChI=1S/C20H15Cl3N2OS.HNO3/c21-14-4-5-16(18(23)8-14)19(9-25-7-6-24-12-25)26-10-13-11-27-20-15(13)2-1-3-17(20)22;2-1(3)4/h1-8,11-12,19H,9-10H2;(H,2,3,4)
InChi Key	HAAITRDZHUANGT-UHFFFAOYSA-N
Canonical SMILES	C1=CC2=C(C(=C1)Cl)SC=C2COC(CN3C=CN=C3)C4=C(C=C(C=C4)Cl)Cl.[N+](=O)(O)[O-]
Isomeric SMILES	C1=CC2=C(C(=C1)Cl)SC=C2COC(CN3C=CN=C3)C4=C(C=C(C=C4)Cl)Cl.[N+](=O)(O)[O-]
WGK Germany	3
PubChem CID	200103
Molecular Weight	500.78

Certificates

Certificate of Analysis(COA)

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7 results found

Lot Number	Certificate Type	Date	Item
D2321186	Certificate of Analysis	Mar 15, 2023	S129395
D2321187	Certificate of Analysis	Mar 15, 2023	S129395
D2321188	Certificate of Analysis	Mar 15, 2023	S129395
D2321192	Certificate of Analysis	Mar 15, 2023	S129395
D2321193	Certificate of Analysis	Mar 15, 2023	S129395
D2321194	Certificate of Analysis	Mar 15, 2023	S129395
D2321195	Certificate of Analysis	Mar 15, 2023	S129395

Solubility

Soluble in DMSO (20 mg/ml), and methanol.

Melt Point(°C)

163-165°C

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