Highly potent and selective δ opioid receptor agonist (K i = 9.4 nM). Centrally active following systemic administration. Displays antidepressant activity.
Storage Temp
Room temperature
Shipped In
Normal
Grade
Moligand™
Action Type
AGONIST
Mechanism of action
Agonist of δ receptor
Note
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour. Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
Product Description
Store at Room Temperature. The product can be stored for up to 12 months.
1.Mann A et al.. (2020) Agonist-induced phosphorylation bar code and differential post-activation signaling of the delta opioid receptor revealed by phosphosite-specific antibodies.. Sci Rep, 10 (8585). [PMID:32444688]
2.Zeng X et al.. (2018) Contribution of TLR4 signaling in intermittent hypoxia-mediated atherosclerosis progression.. J Transl Med, 16 (106). [PMID:29673358]
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