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SP-13786 - 97%, high purity , CAS No.1448440-52-5

1 Citations

≥97%

CAS#: 1448440-52-5
Formula: C₁₇H₁₄F₂N₄O₂
Molecular Weight: 344.32
PubChem CID: 71621488

Item Number

S174266

Grouped product items
SKU	Size	Availability	Price
S174266-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$201.90
S174266-10mg	10mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$297.90
S174266-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$501.90
S174266-50mg	50mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$724.90
S174266-100mg	100mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,016.90

View related series

FAP inhibitor

Basic Description

Synonyms	AKOS027423971 \| EX-A2803 \| N-[2-[(2S)-2-Cyano-4,4-difluoro-1-pyrrolidinyl]-2-oxoethyl]-4-quinolinecarboxamide \| ZB1498 \| S0842 \| PUOOCZVRHBHJRS-NSHDSACASA-N \| A908213 \| AC-36275 \| SB19734 \| DTXSID401131123 \| (S)-N-[2-(2-Cyano-4,4-difluoro-1-pyrrolidinyl)-
Specifications & Purity	≥97%
Storage Temp	Store at 2-8°C,Argon charged
Shipped In	Wet ice

Associated Targets(Human)

FAP Tchem Prolyl endopeptidase FAP (5 Activities)

Discover Target: FAP

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

DPP7 Tchem Dipeptidyl peptidase II (2000 Activities)

Discover Target: DPP7

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

DPP9 Tchem Dipeptidyl peptidase IX (1624 Activities)

Discover Target: DPP9

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

MRC5 (9203 Activities)

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

FAP Tchem Fibroblast activation protein alpha (827 Activities)

Discover Target: FAP

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Liver (3974 Activities)

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Associated Targets(non-human)

DPP4 Dipeptidyl peptidase IV (11 Activities)

Discover Target: DPP4

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

PREP Prolyl endopeptidase (14 Activities)

Discover Target: PREP

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Rattus norvegicus (775804 Activities)

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Fap Seprase (241 Activities)

Discover Target: Fap

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Plasma (328 Activities)

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Liver microsome (341 Activities)

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Names and Identifiers

IUPAC Name	N-[2-[(2S)-2-cyano-4,4-difluoropyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
INCHI	InChI=1S/C17H14F2N4O2/c18-17(19)7-11(8-20)23(10-17)15(24)9-22-16(25)13-5-6-21-14-4-2-1-3-12(13)14/h1-6,11H,7,9-10H2,(H,22,25)/t11-/m0/s1
InChi Key	PUOOCZVRHBHJRS-NSHDSACASA-N
Canonical SMILES	C1C(N(CC1(F)F)C(=O)CNC(=O)C2=CC=NC3=CC=CC=C23)C#N
Isomeric SMILES	C1[C@H](N(CC1(F)F)C(=O)CNC(=O)C2=CC=NC3=CC=CC=C23)C#N
PubChem CID	71621488
Molecular Weight	344.32

Certificates

Certificate of Analysis(COA)

Enter Lot Number to search for COA:

To view the certificate results,please click on a Lot number.For Lot numbers from past orders,please use our order status section

10 results found

Lot Number	Certificate Type	Date	Item
H2414325	Certificate of Analysis	Apr 30, 2024	S174266
H2414326	Certificate of Analysis	Apr 30, 2024	S174266
H2414327	Certificate of Analysis	Apr 30, 2024	S174266
H2414328	Certificate of Analysis	Apr 30, 2024	S174266
H2414329	Certificate of Analysis	Apr 30, 2024	S174266
H2414330	Certificate of Analysis	Apr 30, 2024	S174266
H2414331	Certificate of Analysis	Apr 30, 2024	S174266
H2414332	Certificate of Analysis	Apr 30, 2024	S174266
H2414333	Certificate of Analysis	Apr 30, 2024	S174266
H2414334	Certificate of Analysis	Apr 30, 2024	S174266

Citations of This Product

1. Haiyan Hong, Zhihao Zha, Ruiyue Zhao, Yang Luo, Wenbin Jin, Linlin Li, Ran Wang, Li Yan, Hui Wang, Karl Ploessl, Jinping Qiao, Lin Zhu, Hank F. Kung. (2023) [68Ga]Ga-HBED-CC-FAPI Derivatives with Improved Radiolabeling and Specific Tumor Uptake. MOLECULAR PHARMACEUTICS, 20 (4): (2159–2169). [PMID:36942924]

References

1. Haiyan Hong, Zhihao Zha, Ruiyue Zhao, Yang Luo, Wenbin Jin, Linlin Li, Ran Wang, Li Yan, Hui Wang, Karl Ploessl, Jinping Qiao, Lin Zhu, Hank F. Kung. (2023) [68Ga]Ga-HBED-CC-FAPI Derivatives with Improved Radiolabeling and Specific Tumor Uptake. MOLECULAR PHARMACEUTICS, 20 (4): (2159–2169). [PMID:36942924]

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