JavaScript seems to be disabled in your browser. For the best experience on our site, be sure to turn on Javascript in your browser.

྾

Home
Applications
Targets
G protein-coupled receptors (GPCRs)
Neurotensin receptors
SR48527 , CAS No.156579-04-3, Antagonist of NTS 1 receptor

Skip to the end of the images gallery

Skip to the beginning of the images gallery

SR48527 , CAS No.156579-04-3, Antagonist of NTS 1 receptor

Moligand™

CAS#: 156579-04-3
PubChem CID: 9915499

Item Number

S613697

Grouped product items
SKU	Size	Availability	Price	Qty
S613697-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$625.90
S613697-25mg	25mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,875.90

View related series

NTS1 receptor Antagonist

Basic Description

Synonyms	SR 48527;SR-48527
Specifications & Purity	Moligand™
Grade	Moligand™
Action Type	ANTAGONIST
Mechanism of action	Antagonist of NTS 1 receptor

Associated Targets(Human)

NTSR1 Tchem Neurotensin receptor type 1 (0 Activities)

Discover Target: NTSR1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Associated Targets(non-human)

Ntsr1 Neurotensin receptor 1 (48 Activities)

Discover Target: Ntsr1

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Mechanisms of Action

Mechanism of Action	Action Type	target ID	Target Name	Target Type	Target Organism	Binding Site Name	References

Names and Identifiers

IUPAC Name	(2S)-2-[[1-(7-chloroquinolin-4-yl)-5-(2,6-dimethoxyphenyl)pyrazole-3-carbonyl]amino]-2-cyclohexylacetic acid
INCHI	InChI=1S/C29H29ClN4O5/c1-38-24-9-6-10-25(39-2)26(24)23-16-21(28(35)32-27(29(36)37)17-7-4-3-5-8-17)33-34(23)22-13-14-31-20-15-18(30)11-12-19(20)22/h6,9-17,27H,3-5,7-8H2,1-2H3,(H,32,35)(H,36,37)/t27-/m0/s1
InChi Key	PXNTUYAGLGTUKX-MHZLTWQESA-N
Canonical SMILES	COc1cccc(c1c1cc(nn1c1ccnc2c1ccc(c2)Cl)C(=O)N[C@@H](C1CCCCC1)C(=O)O)OC
Isomeric SMILES	COC1=C(C(=CC=C1)OC)C2=CC(=NN2C3=C4C=CC(=CC4=NC=C3)Cl)C(=O)N[C@@H](C5CCCCC5)C(=O)O
PubChem CID	9915499

Database links

PubChem CID	9915499
ChEMBL Ligand	CHEMBL461604
CAS Registry No.	156579-04-3
GPCRdb Ligand	SR48527

Certificates

Certificate of Analysis(COA)

Enter Lot Number to search for COA:

Solution Calculators

Molarity Calculator

Determine the necessary mass, volume, or concentration for preparing a solution.

Dilution Calculator

Determine the dilution needed to prepare a stock solution.